Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 11708
TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642197(US1184575, 14-acetyl oxycodone)
Affinity DataKi:  18nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642198(US1184575, 6-PEG oxycodone)
Affinity DataKi:  22nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM50370595(US9233167, Oxycodone | Oxycontin | OXYCODONE | US1...)
Affinity DataKi:  30nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642196(US1184575, 6-acetyl oxycodone)
Affinity DataKi:  41nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642199(US1184575, 6,14-bis-PEG oxycodone)
Affinity DataKi:  52nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642200(US1184575, 6-lauroyl oxycodone)
Affinity DataKi:  96nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642201(US1184575, 14-lauroyl oxycodone)
Affinity DataKi:  160nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
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TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandPNGBDBM642202(US1184575, 6,14-bis-lauroyl oxycodone)
Affinity DataKi:  2.22E+4nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
Go to US Patent