Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 12422
TargetHistone deacetylase 3(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM50254780(CHEMBL4078477 | US10301323, Compound D2 | US990889...)
Affinity DataIC50: 43nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 61nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM701605(US12128018, Compound II-234)
Affinity DataIC50: 147nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 1.51E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 2.19E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM50254780(CHEMBL4078477 | US10301323, Compound D2 | US990889...)
Affinity DataIC50: 3.00E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM50254780(CHEMBL4078477 | US10301323, Compound D2 | US990889...)
Affinity DataIC50: 3.35E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM701605(US12128018, Compound II-234)
Affinity DataIC50: 4.45E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM701605(US12128018, Compound II-234)
Affinity DataIC50: 5.14E+3nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 4(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 5(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 7(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 8(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent

TargetHistone deacetylase 9(Human)
Kdac Therapeutics

US Patent
LigandPNGBDBM178100(BRD3308 | US11377423, Cmpd 1 | US12128018, Compoun...)
Affinity DataIC50: 3.00E+4nMAssay Description:Below is a standardized protocol for running HDAC selectivity panel on Caliper LabChip EZ-Reader Instrument.The Caliper HDAC Assay Buffer (acronym HA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2025
Entry Details
Go to US Patent