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Found
181
Enz. Inhib. hit(s) with all data for entry = 13043
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754079
(2-(azepan-1-yl)-5-chloro-4,6-dimethyl-N-(3-sulfamo...)
Copy SMILES
Affinity Data
IC50: 0.700nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754110
(2-(azepan-1-yl)-5-chloro-6-methyl-N-(3-sulfamoylph...)
Copy SMILES
Affinity Data
IC50: 2.10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754160
(2-(6-azaspiro[2.5]- octan-6-yl)-5-chloro- 4,6-dime...)
Copy SMILES
Affinity Data
IC50: 2.20nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754209
(2-[(3S,5R)-4,4- difluoro-3,5-dimethyl- 1-piperidyl...)
Copy SMILES
Affinity Data
IC50: 2.40nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754123
(2-(4,4-difluoroazepan-1-yl)-N-(3-sulfamoylphenyl)-...)
Copy SMILES
Affinity Data
IC50: 2.5nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754243
(5-cyclobutyl-2-(4,4-difluoroazepan-1-yl)-N-(3-sulf...)
Copy SMILES
Affinity Data
IC50: 2.5nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754207
((R or S)-2-(4,4-Difluoro-3-methylpiperidin-1-yl)-N...)
Copy SMILES
Affinity Data
IC50: 3nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754252
(2-(azepan-1-yl)-6-methyl-N-(3-sulfamoylphenyl)-5-(...)
Copy SMILES
Affinity Data
IC50: 3.20nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754245
(5-(but-3-en-1-yl)-2-(4,4-difluoroazepan-1-yl)-N-(3...)
Copy SMILES
Affinity Data
IC50: 3.20nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754089
(2-(azepan-1-yl)-5-chloro- 4,6-dimethyl-N-(3- methy...)
Copy SMILES
Affinity Data
IC50: 3.5nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754090
(6-chloro-2-(4,4- difluoroazepan-1-yl)-4- methyl-N-...)
Copy SMILES
Affinity Data
IC50: 5.80nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754172
(2-(azocan-1-yl)-N-(3- sulfamoylphenyl)-5- (trifluo...)
Copy SMILES
Affinity Data
IC50: 6nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754258
(2-(azepan-1-yl)-6- chloro-4,5-dimethyl-N- (3-sulfa...)
Copy SMILES
Affinity Data
IC50: 6nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM50642031
(US12344595, Example 78)
Copy SMILES
Affinity Data
IC50: 6.10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754093
(6-chloro-2-(4,4- difluoroazepan-1-yl)-N-(3- methyl...)
Copy SMILES
Affinity Data
IC50: 7nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754246
(2-(4,4-difluoroazepan-1-yl)-5-isopropyl-N-(3-sulfa...)
Copy SMILES
Affinity Data
IC50: 7.10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754247
(5-cyclopropyl-2-(4,4- difluoroazepan-1-yl)- N-(3-s...)
Copy SMILES
Affinity Data
IC50: 7.30nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754260
(5-cyano-2-(4,4- difluoroazepan-1-yl)-6- methyl-N-(...)
Copy SMILES
Affinity Data
IC50: 7.30nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754256
(2-(4,4-difluoroazepan-1-yl)-5-(difluoromethoxy)-N-...)
Copy SMILES
Affinity Data
IC50: 7.5nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754083
(2-(azepan-1-yl)-6-chloro- 5-fluoro-4-methyl-N-(3- ...)
Copy SMILES
Affinity Data
IC50: 7.60nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754257
(5-chloro-2-(4,4-difluoroazepan-1-yl)-N-(3-(methyls...)
Copy SMILES
Affinity Data
IC50: 7.80nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754178
(2-(4,4-difluoroazepan-1- yl)-N-(3- methylsulfonylp...)
Copy SMILES
Affinity Data
IC50: 8.40nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754094
(2-(4,4-difluoroazepan-1- yl)-6-methyl-N-(3- methyl...)
Copy SMILES
Affinity Data
IC50: 9.20nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM50642027
(US12344595, Example 44)
Copy SMILES
Affinity Data
IC50: 9.5nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754163
(2-(6- azaspiro[2.6]nonan- 6-yl)-N-(3- sulfamoyl-ph...)
Copy SMILES
Affinity Data
IC50: 10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754113
(2-(azepan-1-yl)-6-chloro-4-methyl-N-(3-sulfamoylph...)
Copy SMILES
Affinity Data
IC50: 10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754241
(2-(azepan-1-yl)-5- cyano-6-methyl-N-(3- sulfamoylp...)
Copy SMILES
Affinity Data
IC50: 10nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754164
(2-(4,4- dimethylazepan-1- yl)-N-(3-sulfamoyl- phen...)
Copy SMILES
Affinity Data
IC50: 11nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754130
(N-(3- sulfamoylphenyl)-2- (4-azatricyclo- [4.3.1.1...)
Copy SMILES
Affinity Data
IC50: 12nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754114
(2-(azepan-1-yl)-5,6- dimethyl-N-(3- sulfamoylpheny...)
Copy SMILES
Affinity Data
IC50: 12nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754129
(2-[rac-3- azabicyclo[3.2.1] octan-3-yl]-N-(3- sulf...)
Copy SMILES
Affinity Data
IC50: 12nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754097
(2-(6-azaspiro[2.5]-octan-6- yl)-N-(3-carbamoyl- ph...)
Copy SMILES
Affinity Data
IC50: 13nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754084
(2-(azepan-1-yl)-4,6- dimethyl-N-(3-sulfamoyl- phen...)
Copy SMILES
Affinity Data
IC50: 14nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754212
(2-[(1R,6R or 1S,6S)- 7,7-difluoro-6-methyl- 3-azab...)
Copy SMILES
Affinity Data
IC50: 14nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754210
(2-[(3S or 3R)-2,2- difluoro-5- azaspiro[2.5]-octan...)
Copy SMILES
Affinity Data
IC50: 14nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754248
(2-(azepan-1-yl)-5-(perfluoroethyl)-N-(3-sulfamoylp...)
Copy SMILES
Affinity Data
IC50: 15nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754229
(2-[(2S,6R)-2-methyl-6- (trifluoromethyl) morpholin...)
Copy SMILES
Affinity Data
IC50: 15nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754208
((R or S)-2-(4,4-Difluoro-3-methylpiperidin-1-yl)-N...)
Copy SMILES
Affinity Data
IC50: 15nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754214
(N-(3- sulfamoylphenyl)-5- (trifluoromethyl)-2- [(1...)
Copy SMILES
Affinity Data
IC50: 16nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754159
(N-(3-carbamoylphenyl)-2-(4,4-difluoroazepan-1-yl)-...)
Copy SMILES
Affinity Data
IC50: 16nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754173
(2-(azepan-1-yl)-6- chloro-N-(3-sulfamoyl- phenyl)p...)
Copy SMILES
Affinity Data
IC50: 16nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754174
(2-(azepan-1-yl)-6- methyl-N-(3-sulfamoyl- phenyl)p...)
Copy SMILES
Affinity Data
IC50: 17nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754098
(N-(3-carbamoyl-phenyl)-6- chloro-2-(4,4- difluoroa...)
Copy SMILES
Affinity Data
IC50: 18nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
TBA
Entry Details
Copy BDB DOI
US Patent
Copy reaction URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754099
(N-(3-carbamoyl-phenyl)-5- chloro-2-(4,4- difluoroa...)
Copy SMILES
Affinity Data
IC50: 19nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
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Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754240
(2-(azepan-1-yl)-5-bromo-6-methoxy-N-(3-sulfamoylph...)
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Affinity Data
IC50: 19nM
Assay Description:
TBD
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In Depth
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Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754179
(2-(azocan-1-yl)-N-(3- methylsulfonylphenyl)- 5-(tr...)
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Affinity Data
IC50: 20nM
Assay Description:
TBD
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In Depth
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Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754217
(N-(3- sulfamoylphenyl)-2- [(1R,5S)-6,6,7,7- tetraf...)
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Affinity Data
IC50: 21nM
Assay Description:
TBD
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Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754115
(2-(azepan-1-yl)-5- chloro-N-(3-sulfamoyl- phenyl)p...)
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Affinity Data
IC50: 22nM
Assay Description:
TBD
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Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754264
(2-cyclopropyl-4-(4,4-difluoroazepan-1-yl)-N-(3-sul...)
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Affinity Data
IC50: 24nM
Assay Description:
TBD
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Merck Sharp & Dohme
US Patent
Ligand
BDBM754100
(N-(3-carbamoyl-phenyl)-5- chloro-2-(4,4-difluoro-1...)
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Affinity Data
IC50: 24nM
Assay Description:
TBD
More data for this Ligand-Target Pair
Target Info
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Ligand Info
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In Depth
Date in BDB:
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