Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 12149
LigandPNGBDBM682742(US20240208953, Example 17A)
Affinity DataIC50: 200nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682741(US20240208953, Example 16B)
Affinity DataIC50: 200nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
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LigandPNGBDBM682740(US20240208953, Example 16A)
Affinity DataIC50: 400nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
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LigandPNGBDBM682754(US20240208953, Example 42B)
Affinity DataIC50: 800nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
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LigandPNGBDBM682745(US20240208953, Example 24C | 6-((R)-2-((3aR,5R,6aS...)
Affinity DataIC50: 1.20E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682743(US20240208953, Example 18B)
Affinity DataIC50: 1.20E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682739(US20240208953, Example 14B)
Affinity DataIC50: 1.30E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682738(US20240208953, Example 10A)
Affinity DataIC50: 2.10E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682753(US20240208953, Example 42A)
Affinity DataIC50: 2.20E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682746(US20240208953, Example 28A | 6-((R)-1-hydroxy-2-((...)
Affinity DataIC50: 2.40E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682737(US20240208953, Example 8A)
Affinity DataIC50: 2.80E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682744(US20240208953, Example 21)
Affinity DataIC50: 3.60E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682749(US20240208953, Example 31B | 8-fluoro-6-((S)-1-hyd...)
Affinity DataIC50: 3.90E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682751(US20240208953, Example 33B)
Affinity DataIC50: 4.90E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682752(US20240208953, Example 36A)
Affinity DataIC50: 5.50E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682734(US20240208953, Example 5D)
Affinity DataIC50: 5.90E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682733(US20240208953, Example 5C)
Affinity DataIC50: 6.00E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682748(US20240208953, Example 31A | 8-fluoro-6-((R)-1-hyd...)
Affinity DataIC50: 7.30E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682731(US20240208953, Example 1B | 6-((S)-1-hydroxy-2-((3...)
Affinity DataIC50: 7.60E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682746(US20240208953, Example 28A | 6-((R)-1-hydroxy-2-((...)
Affinity DataIC50: 8.20E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682732(US20240208953, Example 4B | 6-((S)-2-((3aS,4S,5S,6...)
Affinity DataIC50: 9.20E+3nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682730(US20240208953, Example 1A | 6-((R)-1-hydroxy-2-((3...)
Affinity DataIC50: 1.07E+4nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
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LigandPNGBDBM682747(US20240208953, Example 29B | 8-fluoro-6-((S)-2-((3...)
Affinity DataIC50: 1.25E+4nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682735(US20240208953, Example 6C | 8-fluoro-6-((R)-2-((3a...)
Affinity DataIC50: 1.33E+4nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682736(US20240208953, Example 7B)
Affinity DataIC50: 1.52E+4nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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LigandPNGBDBM682755(US20240208953, Example 44B | (3aS,4S,5S,6aR)-5-(2-...)
Affinity DataIC50: 1.57E+4nMAssay Description:hERG currents were recorded using the Qpatch automated patch clamp systems (Sophion Bioscience Inc., North Brunswick, NJ) in the whole (single) cell ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
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