Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 12391
LigandPNGBDBM700200(1-[[2- (difluoromethoxy)pyridin- 4-yl]methyl]-3- [...)
Affinity DataEC50:  230nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700187(US20240336571, Example 28 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  1.36E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700188(US20240336571, Example 29 | 1-[(1S)-1-(2- methoxyp...)
Affinity DataEC50:  520nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700189(US20240336571, Example 30 | 1-((S)-1-(2- (difluoro...)
Affinity DataEC50:  210nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700190(US20240336571, Example 31 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  500nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700191(US20240336571, Example 32 | 1-[2-(oxetan-3- yl)pyr...)
Affinity DataEC50:  3.02E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700192(US20240336571, Example 33 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  310nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700193(US20240336571, Example 34 | 1-[(2-phenoxypyridin- ...)
Affinity DataEC50:  4.78E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700194(US20240336571, Example 35 | 1-[[2-(2,2- difluoroet...)
Affinity DataEC50:  200nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700195(US20240336571, Example 36 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  120nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700196(US20240336571, Example 37 | 1-[2- (fluoromethoxy)p...)
Affinity DataEC50:  910nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700197(US20240336571, Example 38 | 1-[1-[2- (difluorometh...)
Affinity DataEC50:  3.81E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700198(US20240336571, Example 39 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  70nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700199(US20240336571, Example 40 | 1-[rac-(1R,2S)-2- cycl...)
Affinity DataEC50:  780nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700186(US20240336571, Example 27 | 1-[(2-imidazol-1- ylpy...)
Affinity DataEC50:  2.84E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700201(US20240336571, Example 42 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  1.03E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700202(US20240336571, Example 43 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  8.01E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700203(US20240336571, Example 44 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  330nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700204(US20240336571, Example 45 | 1-(2- cyclohexylcyclop...)
Affinity DataEC50:  880nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700205(US20240336571, Example 46 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  900nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700206(US20240336571, Example 47 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  50nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700207(US20240336571, Example 48 | 1-[[2-(2,3- difluoropr...)
Affinity DataEC50:  570nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700208(US20240336571, Example 49 | 1-[[2- (difluoromethox...)
Affinity DataEC50:  3.83E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700200(1-[[2- (difluoromethoxy)pyridin- 4-yl]methyl]-3- [...)
Affinity DataEC50:  620nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700210(US20240336571, Example 51 | 1-[rac-(1R,2R)-2- (tri...)
Affinity DataEC50:  280nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700211(US20240336571, Example 52 | 1-[[6- (difluoromethox...)
Affinity DataEC50:  1.00E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700212(US20240336571, Example 53 | 1-[[2-[(2R)-1,1,1- tri...)
Affinity DataEC50:  360nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700173(US20240336571, Example 14 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  70nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700161(US20240336571, Example 2 | 1-[rac-(1R,2S)-2- cyclo...)
Affinity DataEC50:  570nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700162(US20240336571, Example 3 | 1-[(6-chloropyridin-2- ...)
Affinity DataEC50:  1.54E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700163(US20240336571, Example 4 | 1-[(2-propan-2- ylpyrim...)
Affinity DataEC50:  4.40E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700164(BDBM700168 | 1-[(2-methoxypyridin- 4-yl)methyl]-3-...)
Affinity DataEC50:  3.75E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700165(US20240336571, Example 6 | 1-[(1R,2S)-2- phenylcyc...)
Affinity DataEC50:  660nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700166(US20240336571, Example 7 | 1-[[2- (difluoromethoxy...)
Affinity DataEC50:  100nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700167(BDBM700169 | 1-[(2-cyanopyridin-4- yl)methyl]-3-[r...)
Affinity DataEC50:  4.18E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700164(BDBM700168 | 1-[(2-methoxypyridin- 4-yl)methyl]-3-...)
Affinity DataEC50:  3.41E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700167(BDBM700169 | 1-[(2-cyanopyridin-4- yl)methyl]-3-[r...)
Affinity DataEC50:  1.19E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700170(US20240336571, Example 11 | 1-(2- cyclohexylcyclop...)
Affinity DataEC50:  2.14E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700171(1-[(2-pyrazol-1- ylpyridin-4-yl)methyl]- 3-[rac-(1...)
Affinity DataEC50:  670nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700171(1-[(2-pyrazol-1- ylpyridin-4-yl)methyl]- 3-[rac-(1...)
Affinity DataEC50:  1.34E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700160(US20240336571, Example 1 | 1-[(4-cyanopyridin-2- y...)
Affinity DataEC50:  4.68E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700174(US20240336571, Example 15 | 1-[(1S,2R)-2- cyclohex...)
Affinity DataEC50:  1.57E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700175(US20240336571, Example 16 | 1-[2-(oxetan-3- yloxy)...)
Affinity DataEC50:  960nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700176(US20240336571, Example 17 | 1-[(2-chloropyridin-4-...)
Affinity DataEC50:  1.76E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700177(US20240336571, Example 18 | 1-[(6-cyanopyridin-2- ...)
Affinity DataEC50:  3.02E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700178(US20240336571, Example 19 | 1-[(2-chloropyridin-4-...)
Affinity DataEC50:  6.83E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700179(US20240336571, Example 20 | 1-[[2-(oxan-4- yloxy)p...)
Affinity DataEC50:  5.93E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700180(US20240336571, Example 21 | 1-[[2- (difluoromethyl...)
Affinity DataEC50:  3.20E+3nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700181(US20240336571, Example 22 | 1-[(1R,2S)-2- phenylcy...)
Affinity DataEC50:  720nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700182(US20240336571, Example 23 | 1-[[2-(1,3-oxazol-5- y...)
Affinity DataEC50:  920nMAssay Description:At the beginning of each assay, 20 μl of cell suspension was dispensed into each well of a multi-hole 384-well SyncroPatch chip by the onboard p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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