Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 12393
LigandPNGBDBM700285(Dimethyl-oxo-[[2-[[4-[4-(4-pyridyl)-1H-pyrazol-3-y...)
Affinity DataIC50: 0.0500nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700280(N-[Dimethyl(oxo)-lambda6- sulfanylidene]-2-[[4- [1...)
Affinity DataIC50: 0.0630nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700283(2-[[4-[4-(4-Pyridyl)-1H-pyrazol-3-yl]phenoxy]methy...)
Affinity DataIC50: 0.0630nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700235(N-[Dimethyl(oxo)-λ6-sulfanylidene]-2-[[4-[4-(...)
Affinity DataIC50: 0.0630nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700215(2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]phenoxy]...)
Affinity DataIC50: 0.0790nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700216(Ammonium 2-[[4-[1-methyl-4-(4-pyridyl)pyrazol-3-yl...)
Affinity DataIC50: 0.0790nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700291(4-[2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]pheno...)
Affinity DataIC50: 0.0790nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700244(2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]phenoxy]...)
Affinity DataIC50: 0.0790nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700249(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-2- [[4-[1...)
Affinity DataIC50: 0.0790nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700282(2-[[4-[4-(4-Pyridyl)-1H-pyrazol-3-yl]phenoxy]methy...)
Affinity DataIC50: 0.100nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700248(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-2- [4-[1-...)
Affinity DataIC50: 0.100nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700284(N-[Dimethyl(oxo)-λ6-sulfanylidene]-2-[[4-[4-(...)
Affinity DataIC50: 0.100nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700252(N-(Cyclopropyl- methyl-oxo-lambda6- sulfanylidene)...)
Affinity DataIC50: 0.100nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700257(N-[Dimethyl(oxo)-λ6-sulfanylidene]-2-[[4-[1-m...)
Affinity DataIC50: 0.120nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700256(N-Methyl-2-[[4-[1-methyl-4-(4-pyridyl)pyrazol-3-yl...)
Affinity DataIC50: 0.135nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700251(2-[[4-[1-Methyl-4-(4- pyridyl)pyrazol-3- yl]phenox...)
Affinity DataIC50: 0.138nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700250(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-2- [[4-[4...)
Affinity DataIC50: 0.145nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700263(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-2- [[4-[1...)
Affinity DataIC50: 0.174nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700214(2-[[4-[2-Methyl-4-(4-pyridyl)pyrazol-3-yl]phenoxy]...)
Affinity DataIC50: 0.204nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700288(1-Methyl-3-[2-[[4-[1-methyl-4-(4-pyridyl)pyrazol-3...)
Affinity DataIC50: 0.214nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700233(N-[Dimethyl(oxo)-λ6-sulfanylidene]-5-methyl-2...)
Affinity DataIC50: 0.224nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700290(4-[2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]pheno...)
Affinity DataIC50: 0.224nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700269(N-[Dimethyl(oxo)-lambda6- sulfanylidene]-5- fluoro...)
Affinity DataIC50: 0.257nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700287(N-[2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]pheno...)
Affinity DataIC50: 0.288nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700268(N-[Dimethyl(oxo)-lambda6- sulfanylidene]-6- fluoro...)
Affinity DataIC50: 0.324nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700292(1-[2-[[4-[1-Methyl-4-(4-pyridyl)pyrazol-3-yl]pheno...)
Affinity DataIC50: 0.347nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700289(1-[Dimethyl(oxo)-λ6-sulfanylidene]-3-[2-[[4-[...)
Affinity DataIC50: 0.347nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700294(1-[3-[[4-[1-Methyl-4- (4-pyridyl)pyrazol- 3- yl]ph...)
Affinity DataIC50: 0.355nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700213(2-[[4-[2-Methyl-4-(4-pyridyl)pyrazol-3-yl]phenoxy]...)
Affinity DataIC50: 0.372nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700261(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-2- [[4-[1...)
Affinity DataIC50: 0.372nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700281(2-[[4-[1-Cyclopropyl- 4-(4-pyridyl)pyrazol- 3- yl]...)
Affinity DataIC50: 0.380nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700278(N-[Dimethyl(oxo)-lambda6- sulfanylidene]-6- fluoro...)
Affinity DataIC50: 0.389nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700217(2-[4-(4-Pyridyl)-3-[4-(2-quinolylmethoxy)phenyl]py...)
Affinity DataIC50: 0.389nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700258(N-[Dimethyl(oxo)- lambda6-sulfanylidene]-3- [[4-[1...)
Affinity DataIC50: 0.457nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700286(Imino-methyl-oxo-[2-[[4-[4-(4-pyridyl)-1H-pyrazol-...)
Affinity DataIC50: 0.479nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700255(N-Methyl-2-[[4-[1-methyl-4-(4-pyridyl)pyrazol-3-yl...)
Affinity DataIC50: 0.603nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700279(5-Chloro-N- [Dimethyl(oxo)-lambda6- sulfanylidene]...)
Affinity DataIC50: 0.741nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700293(2-[[4-[1-Methyl-4-(4- pyridyl)pyrazol-3- yl]phenox...)
Affinity DataIC50: 1.05nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700295(2-[[4-[1-Methyl-4-(4- pyridyl)pyrazol-3- yl]phenox...)
Affinity DataIC50: 1.10nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700218(2-[[4-[1-Methylsulfonyl-4-(4-pyridyl)pyrazol-3-yl]...)
Affinity DataIC50: 4.37nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700264(N-[Dimethyl(oxo)-λ6-sulfanylidene]-7-fluoro-2...)
Affinity DataIC50: 4.79nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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LigandPNGBDBM700272(N-[Dimethyl(oxo)-lambda6- sulfanylidene]-6- methyl...)
Affinity DataIC50: 5.13nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2025
Entry Details
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