Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 12471
TargetAdenosine receptor A2a(Human)
Shanghai Haiyan Pharmaceutical Technology Co.

US Patent
LigandPNGBDBM704701(US20240376081, Compound X)
Affinity DataIC50: 24nMAssay Description:The screening procedure was as follows:1. adjusting the cell density to 6×105 cells/mL with serum-free medium;2. adding 5 mL of cytosol, 2.5 mL of NE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Shanghai Haiyan Pharmaceutical Technology Co.

US Patent
LigandPNGBDBM704701(US20240376081, Compound X)
Affinity DataIC50: 62nMAssay Description:The screening procedure was as follows:1. adjusting the cell density to 6×105 cells/mL with serum-free medium;2. adding 5 mL of cytosol, 2.5 mL of NE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetAdenosine receptor A2a(Human)
Shanghai Haiyan Pharmaceutical Technology Co.

US Patent
LigandPNGBDBM50594625(Etrumadenant | Ab-928 | Ab928 | AB-928 | AB928 | E...)
Affinity DataIC50: 65nMAssay Description:The screening procedure was as follows:1. adjusting the cell density to 6×105 cells/mL with serum-free medium;2. adding 5 mL of cytosol, 2.5 mL of NE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetAdenosine receptor A2b(Human)
Shanghai Haiyan Pharmaceutical Technology Co.

US Patent
LigandPNGBDBM50594625(Etrumadenant | Ab-928 | Ab928 | AB-928 | AB928 | E...)
Affinity DataIC50: 75nMAssay Description:The screening procedure was as follows:1. adjusting the cell density to 6×105 cells/mL with serum-free medium;2. adding 5 mL of cytosol, 2.5 mL of NE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent