Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 12474
TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704883(US20240376093, Compound 3)
Affinity DataIC50: 0.0300nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704881(US20240376093, Compound 1)
Affinity DataIC50: 0.0400nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704892(US20240376093, Compound 12)
Affinity DataIC50: 0.0500nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704882(US20240376093, Compound 2)
Affinity DataIC50: 0.0600nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704890(US20240376093, Compound 10)
Affinity DataIC50: 0.0600nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704884(US20240376093, Compound 4)
Affinity DataIC50: 0.0700nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704885(US20240376093, Compound 5)
Affinity DataIC50: 0.0700nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704889(US20240376093, Compound 9)
Affinity DataIC50: 0.0700nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704896(US20240376093, Compound 16)
Affinity DataIC50: 0.0800nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704895(US20240376093, Compound 15)
Affinity DataIC50: 0.0800nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704887(US20240376093, Compound 7)
Affinity DataIC50: 0.0900nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704904(US20240376093, Compound 27)
Affinity DataIC50: 0.0900nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704898(US20240376093, Compound 18)
Affinity DataIC50: 0.0900nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704891(US20240376093, Compound 11)
Affinity DataIC50: 0.110nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704906(US20240376093, Compound 29)
Affinity DataIC50: 0.110nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704893(US20240376093, Compound 13)
Affinity DataIC50: 0.120nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704899(US20240376093, Compound 19)
Affinity DataIC50: 0.120nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704903(US20240376093, Compound 23)
Affinity DataIC50: 0.130nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704901(US20240376093, Compound 21)
Affinity DataIC50: 0.130nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704902(US20240376093, Compound 22)
Affinity DataIC50: 0.140nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704888(US20240376093, Compound 8)
Affinity DataIC50: 0.150nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704905(US20240376093, Compound 28)
Affinity DataIC50: 0.170nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704886(US20240376093, Compound 6)
Affinity DataIC50: 0.180nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704900(US20240376093, Compound 20)
Affinity DataIC50: 0.190nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704894(US20240376093, Compound 14)
Affinity DataIC50: 0.25nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704897(US20240376093, Compound 17)
Affinity DataIC50: 0.290nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704910(US20240376093, Compound 33)
Affinity DataIC50: 0.300nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704909(US20240376093, Compound 32)
Affinity DataIC50: 0.310nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704908(US20240376093, Compound 31)
Affinity DataIC50: 0.340nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704907(US20240376093, Compound 30)
Affinity DataIC50: 0.560nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2 [575-869](Human)
Medshine Discovery

US Patent
LigandPNGBDBM704911(US20240376093, Compound 35)
Affinity DataIC50: 0.760nMAssay Description:0.5 nM TYK2 protein (His-TVMV-TYK2 JH2 (575-869)), 0.2 nM terbium-labeled His antibody, fluorescein-labeled kinase tracer at the relevant Kd value, a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/20/2025
Entry Details
Go to US Patent