Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 12585
TargetHistone-lysine N-methyltransferase, H3 lysine-36 specific(Human)
K36 Therapeutics

US Patent
LigandPNGBDBM712326(US20250011329, Compound III-35)
Affinity DataIC50: 1nMAssay Description:A reaction mixture was prepared by adding oligonucleosomes from Chicken (0.05 mg/ml) to freshly prepared reaction buffer containing 50 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
Go to US Patent

TargetHistone-lysine N-methyltransferase NSD2(Human)
K36 Therapeutics

US Patent
LigandPNGBDBM712326(US20250011329, Compound III-35)
Affinity DataIC50: 2nMAssay Description:A reaction mixture was prepared by adding oligonucleosomes from Chicken (0.05 mg/ml) to freshly prepared reaction buffer containing 50 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
Go to US Patent

TargetHistone-lysine N-methyltransferase NSD2(Human)
K36 Therapeutics

US Patent
LigandPNGBDBM712321(US20250011329, Compound J)
Affinity DataIC50: 11nMAssay Description:A reaction mixture was prepared by adding oligonucleosomes from Chicken (0.05 mg/ml) to freshly prepared reaction buffer containing 50 mM Tris-HCl (p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
Go to US Patent