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Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 13241
TargetEpidermal growth factor receptor(Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770153(23-[(3-fluoro-2-methoxyphenyl)amino]-8,11- dioxa-5...)
Affinity DataEC50: <1nMAssay Description:Table D: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor [1-770,'NPG',771-1210,T790M](Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770154((13Z)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50: <1nMAssay Description:Table B: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770154((13Z)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table D: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770155((16R)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table D: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770156((16S)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table D: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor [1-770,'NPG',771-1210,T790M](Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770152((13E)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table B: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor [1-770,'NPG',771-1210,T790M](Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770153(23-[(3-fluoro-2-methoxyphenyl)amino]-8,11- dioxa-5...)
Affinity DataEC50:  3nMAssay Description:Table B: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor [1-770,'NPG',771-1210,T790M](Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770155((16R)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table B: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor [1-770,'NPG',771-1210,T790M](Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770156((16S)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table B: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent

TargetEpidermal growth factor receptor(Human)
Celyn Therapeutics

US Patent
LigandPNGBDBM770152((13E)-23-[(3-fluoro-2- methoxyphenyl)amino]-8,11-d...)
Affinity DataEC50:  3nMAssay Description:Table D: The enzymatic assay used to determine activity was a Luminescence assay using a Microplate Reader ClarioStar Plus. The enzymatic reaction wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/22/2025
Entry Details
US Patent