Compile Data Set for Download or QSAR
Report error Found 258 Enz. Inhib. hit(s) with all data for entry = 13403
TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787121BDBM787121((2S)-3-amino-2-benzyl-N-[3-(1H-pyrazol-4-yl)-1H-in...)
Affinity DataIC50: 0.0900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787109BDBM787109(Preparation of (2R)-2-amino-2-(3-methoxyphenyl)-N-...)
Affinity DataIC50: 0.100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787093BDBM787093(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-cy...)
Affinity DataIC50: 0.130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787082BDBM787082(Preparation of (2S)-2-amino-2-phenyl-N-[3-(1H-pyra...)
Affinity DataIC50: 0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787088BDBM787088(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(3...)
Affinity DataIC50: 0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787077BDBM787077(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(4...)
Affinity DataIC50: 0.170nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787154BDBM787154(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(m...)
Affinity DataIC50: 0.180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787107BDBM787107(US20250346616, Example 40)
Affinity DataIC50: 0.180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787147BDBM787147(3-amino-2-(4-aminophenyl)-N-[3-(1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 0.180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787109BDBM787109(Preparation of (2R)-2-amino-2-(3-methoxyphenyl)-N-...)
Affinity DataIC50: 0.180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787121BDBM787121((2S)-3-amino-2-benzyl-N-[3-(1H-pyrazol-4-yl)-1H-in...)
Affinity DataIC50: 0.180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787131BDBM787131(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(3...)
Affinity DataIC50: 0.190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787093BDBM787093(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-cy...)
Affinity DataIC50: 0.190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787171BDBM787171(2-[4-(2-aminoethyl) piperazin-1-yl]-2-phenyl-N-[3-...)
Affinity DataIC50: 0.220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787117BDBM787117(3-(1-((3-(1H-pyrazol-4-yl)-1H-indol-7-yl)amino)-3-...)
Affinity DataIC50: 0.220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787082BDBM787082(Preparation of (2S)-2-amino-2-phenyl-N-[3-(1H-pyra...)
Affinity DataIC50: 0.240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787130BDBM787130(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(5...)
Affinity DataIC50: 0.240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787100BDBM787100(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(p...)
Affinity DataIC50: 0.240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787190BDBM787190(N-(2-amino-1-(3-methoxyphenyl)ethyl)-3-(1H-pyrazol...)
Affinity DataIC50: 0.240nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787105BDBM787105(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-(4-methylp...)
Affinity DataIC50: 0.260nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787076BDBM787076(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(4...)
Affinity DataIC50: 0.270nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787112BDBM787112(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-2-(1-methylp...)
Affinity DataIC50: 0.270nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787154BDBM787154(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(m...)
Affinity DataIC50: 0.290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787088BDBM787088(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(3...)
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787117BDBM787117(3-(1-((3-(1H-pyrazol-4-yl)-1H-indol-7-yl)amino)-3-...)
Affinity DataIC50: 0.320nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787107BDBM787107(US20250346616, Example 40)
Affinity DataIC50: 0.330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787077BDBM787077(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(4...)
Affinity DataIC50: 0.330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787131BDBM787131(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(3...)
Affinity DataIC50: 0.370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787086BDBM787086(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(3...)
Affinity DataIC50: 0.370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787186BDBM787186(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-2-amino-2-(p...)
Affinity DataIC50: 0.390nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787147BDBM787147(3-amino-2-(4-aminophenyl)-N-[3-(1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 0.390nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787201BDBM787201(N-(1-amino-3-phenylpropan-2-yl)-3-(1H-pyrazol-4-yl...)
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787171BDBM787171(2-[4-(2-aminoethyl) piperazin-1-yl]-2-phenyl-N-[3-...)
Affinity DataIC50: 0.420nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787130BDBM787130(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(5...)
Affinity DataIC50: 0.430nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787104BDBM787104(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-(4-methylp...)
Affinity DataIC50: 0.430nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787105BDBM787105(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-(4-methylp...)
Affinity DataIC50: 0.440nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787177BDBM787177(4-(1-((3-(1H-pyrazol-4-yl)-1H-indol-7-yl)amino)-3-...)
Affinity DataIC50: 0.470nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787099BDBM787099(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(p...)
Affinity DataIC50: 0.480nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787152BDBM787152(3-amino-2-(4-fluorophenyl)-N-[3-(1H-pyrazol-4-yl)-...)
Affinity DataIC50: 0.520nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787169BDBM787169(3-amino-2-(1-methyl-2-oxopyridin-4-yl)-N-[3-(1H-py...)
Affinity DataIC50: 0.530nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787112BDBM787112(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-2-(1-methylp...)
Affinity DataIC50: 0.530nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787100BDBM787100(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(p...)
Affinity DataIC50: 0.550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787168BDBM787168(3-amino-2-(5-methoxypyridin-3-yl)-N-[3-(1H-pyrazol...)
Affinity DataIC50: 0.560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787076BDBM787076(N-(3-(1H-pyrazol-4-yl)-1H-indol-7-yl)-3-amino-2-(4...)
Affinity DataIC50: 0.590nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787119BDBM787119(3-amino-2-benzyl-N-[3-(1H-pyrazol-4-yl)-1H-indol-7...)
Affinity DataIC50: 0.590nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787137BDBM787137(3-(2-amino-1-{[3-(1H-pyrazol-4-yl)-1H-indol-7-yl]c...)
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787141BDBM787141(4-(1-((3-(1H-pyrazol-4-yl)-1H-indol-7-yl)amino)-3-...)
Affinity DataIC50: 0.620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787190BDBM787190(N-(2-amino-1-(3-methoxyphenyl)ethyl)-3-(1H-pyrazol...)
Affinity DataIC50: 0.620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787083BDBM787083([4-[(1S)-1-(aminomethyl)-2-oxo-2-[[3-(1H-pyrazol-4...)
Affinity DataIC50: 0.630nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Dizal (Jiangsu) Pharmaceutical Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 787204BDBM787204(Preparation of (2S)-3-amino-2-phenyl-N-[7-(1H-pyra...)
Affinity DataIC50: 0.630nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/5/2026
Entry Details
US Patent

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