Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 5854
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:Syk was pre-activated at room temperature for 30 mins in the presence of 16.6 mM MgCl2, 8.3 mM ATP and then diluted to 4 nM in 40 mM Hepes pH 7.4, 0....More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 7.90E+3nMpH: 7.5 T: 2°CAssay Description:VEGFR2 (100 nM typically) was activated at room temperature for 20 min. in the presence of 100 mM HEPES, pH 7.5, 10 mM MgCl2, 100 μM ATP, 300 μ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMpH: 8.0 T: 2°CAssay Description:Aurora B (2 μM) was preactivated by equivalent concentration of GST-INCENP in 30 mM Tris-HCl pH 8.0, 0.4 mM ATP, 2 mM MgCl2, 0.1 mM EGTA, 0.1% BME...More data for this Ligand-Target Pair
