Compile Data Set for Download or QSAR
Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 6145
Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111790(US8618114, 1.2.22(5).HCl)
Affinity DataIC50: 0.227nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111771(US8618114, 1.2.11(1))
Affinity DataIC50: 0.293nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417932(CHEMBL1668587 | US8618114, 1.2.4(1))
Affinity DataIC50: 0.340nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111787(US8618114, 1.2.22(2).HCl)
Affinity DataIC50: 0.560nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111788(US8618114, 1.2.22(3).HCl)
Affinity DataIC50: 0.645nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111785(US8618114, 1.2.22(1).HCl)
Affinity DataIC50: 0.670nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417915(CHEMBL1668586 | US8618114, 1.2.3(1))
Affinity DataIC50: 0.740nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417933(CHEMBL1668588 | US8618114, 1.2.7(1))
Affinity DataIC50: 0.880nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111780(US8618114, 1.2.13(3))
Affinity DataIC50: 1.28nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417915(CHEMBL1668586 | US8618114, 1.2.3(1))
Affinity DataIC50: 3nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417916(CHEMBL1668564 | US8618114, 1.2.5(1))
Affinity DataIC50: 4nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111767(US8618114, 1.2.8(8))
Affinity DataIC50: 4nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417917(CHEMBL1668565 | US8618114, 1.2.6(1))
Affinity DataIC50: 4nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111775(US8618114, 1.2.12(4).HCl)
Affinity DataIC50: 4.19nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417918(CHEMBL1668589 | US8618114, 1.2.1(4))
Affinity DataIC50: 5.01nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111787(US8618114, 1.2.22(2).HCl)
Affinity DataIC50: 9nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111772(US8618114, 1.2.19(2).HCl)
Affinity DataIC50: 9nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111770(US8618114, 1.2.10(3))
Affinity DataIC50: 10nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111756(US8618114, 1.1(4))
Affinity DataIC50: 10nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111790(US8618114, 1.2.22(5).HCl)
Affinity DataIC50: 10nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111764(US8618114, 1.1.8(3))
Affinity DataIC50: 10nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
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Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111764(US8618114, 1.1.8(3))
Affinity DataIC50: 10nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111785(US8618114, 1.2.22(1).HCl)
Affinity DataIC50: 11.3nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111773(US8618114, 1.2.12(2))
Affinity DataIC50: 12nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111771(US8618114, 1.2.11(1))
Affinity DataIC50: 12nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111770(US8618114, 1.2.10(3))
Affinity DataIC50: 12nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111781(US8618114, 1.2.19(1).CH3CO2H)
Affinity DataIC50: 15.3nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417914(CHEMBL1668585 | US8618114, 1.2.2(1))
Affinity DataIC50: 16nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417935(CHEMBL1668593 | US8618114, 1.2.1(2))
Affinity DataIC50: 18nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417933(CHEMBL1668588 | US8618114, 1.2.7(1))
Affinity DataIC50: 19nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111794(US8618114, 1.2.22(11).HCl)
Affinity DataIC50: 22nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417918(CHEMBL1668589 | US8618114, 1.2.1(4))
Affinity DataIC50: 24nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111791(US8618114, 1.2.22(6).HCl)
Affinity DataIC50: 25.2nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111792(US8618114, 1.2.22(10).HCl)
Affinity DataIC50: 26nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111776(US8618114, 1.1.12(5))
Affinity DataIC50: 31.0nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417924(CHEMBL1668502 | US8618114, 1.1.3(1))
Affinity DataIC50: 40nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417935(CHEMBL1668593 | US8618114, 1.2.1(2))
Affinity DataIC50: 45nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111788(US8618114, 1.2.22(3).HCl)
Affinity DataIC50: 45nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111761(US8618114, 1.1.2(2))
Affinity DataIC50: 50nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111758(US8618114, 1.1(6))
Affinity DataIC50: 50nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111757(US8618114, 1.1(5))
Affinity DataIC50: 50nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111765(US8618114, 1.2(1))
Affinity DataIC50: 52nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111797(US8618114, 1.2.22(14).HCl)
Affinity DataIC50: 56.4nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111774(US8618114, 1.2.12(3))
Affinity DataIC50: 69.9nMAssay Description:Screening of the disclosed compounds for their potential ability to interact with serotonin 5-HT6 receptors was carried out by method of radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417904(CHEMBL1668568 | US8618114, 1.1.6(1))
Affinity DataIC50: 73nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417913(CHEMBL1668583 | US8618114, 1.2.1(1))
Affinity DataIC50: 76nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111789(US8618114, 1.2.22(4).HCl)
Affinity DataIC50: 78nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM50417932(CHEMBL1668587 | US8618114, 1.2.4(1))
Affinity DataIC50: 101nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111762(US8618114, 1.1.3(5))
Affinity DataIC50: 156nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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Target5-hydroxytryptamine receptor 6(Human)
TBA

US Patent
LigandPNGBDBM111778(US8618114, 1.2.12(12) | US8618114, 1.2.12(11))
Affinity DataIC50: 172nMAssay Description:Determination of antagonistic activity of compounds of the general formula 1 towards 5-HT6 receptors. Compounds of the general formula 1 were tested ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2014
Entry Details
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