Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 6376
LigandPNGBDBM125036(US8772510, 55)
Affinity DataIC50: 0.390nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125038(US8772510, 57)
Affinity DataIC50: 0.470nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125040(US8772510, 59 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.530nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125041(US8772510, 60 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.670nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125039(US8772510, 58)
Affinity DataIC50: 0.700nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125012(US8772510, 31 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 1.70nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125046(US8772510, 65 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 1.83nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125013(US8772510, 32 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.10nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125037(US8772510, 56 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.41nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125026(US8772510, 45 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.70nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125017(US8772510, 36 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.77nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124988(US8772510, 7)
Affinity DataIC50: 4nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125016(US8772510, 35 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 5.66nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125043(US8772510, 62 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 7.41nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125008(US8772510, 27 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 11nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125005(US8772510, 24)
Affinity DataIC50: 12.4nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124985(US8772510, 4)
Affinity DataIC50: 13.4nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125021(US8772510, 40)
Affinity DataIC50: 13.8nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125001(US8772510, 20)
Affinity DataIC50: 14.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125028(US8772510, 47)
Affinity DataIC50: 14.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124983(US8772510, 2)
Affinity DataIC50: 16nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125024(US8772510, 43)
Affinity DataIC50: 16.8nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125020(US8772510, 39)
Affinity DataIC50: 18.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125009(US8772510, 28)
Affinity DataIC50: 19.3nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124997(US8772510, 16)
Affinity DataIC50: 20.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125003(US8772510, 22)
Affinity DataIC50: 21.3nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125007(US8772510, 26)
Affinity DataIC50: 23.8nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125019(US8772510, 38)
Affinity DataIC50: 27.3nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125034(US8772510, 53)
Affinity DataIC50: 31nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125010(US8772510, 29)
Affinity DataIC50: 32.8nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124992(US8772510, 11)
Affinity DataIC50: 34.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125011(US8772510, 30 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 38.5nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125030(US8772510, 49 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 44.9nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125018(US8772510, 37)
Affinity DataIC50: 45.9nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125042(US8772510, 61 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 54.2nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125044(US8772510, 63 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 56.9nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124984(US8772510, 3)
Affinity DataIC50: 64nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
Entry Details
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LigandPNGBDBM124993(US8772510, 12)
Affinity DataIC50: 73nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125033(US8772510, 52 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 73.7nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125004(US8772510, 23)
Affinity DataIC50: 77.9nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125014(US8772510, 33 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 86nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124982(US8772510, 1)
Affinity DataIC50: 86.6nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124999(US8772510, 18)
Affinity DataIC50: 110nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125025(US8772510, 44)
Affinity DataIC50: 136nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125032(US8772510, 51)
Affinity DataIC50: 145nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM125035(US8772510, 54)
Affinity DataIC50: 180nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
Entry Details
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LigandPNGBDBM124990(US8772510, 9)
Affinity DataIC50: 189nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
Entry Details
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LigandPNGBDBM125002(US8772510, 21)
Affinity DataIC50: 202nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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LigandPNGBDBM124996(US8772510, 15)
Affinity DataIC50: 207nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
Entry Details
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LigandPNGBDBM125000(US8772510, 19)
Affinity DataIC50: 225nMAssay Description:PDE10 activity of the compounds of the present invention was determined using a Scintillation Proximity Assay (SPA)-based method similar to the one p...More data for this Ligand-Target Pair
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Date in BDB:
11/24/2014
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