Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 7028
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167443(US9073906, 128)
Affinity DataIC50: 0.100nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167438(US9073906, 88)
Affinity DataIC50: 0.200nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167440(US9073906, 122)
Affinity DataIC50: 0.400nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167441(US9073906, 123)
Affinity DataIC50: 0.800nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167444(US9073906, 156)
Affinity DataIC50: 1nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167451(US9073906, 196)
Affinity DataIC50: 1.30nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167437(US9073906, 69)
Affinity DataIC50: 3nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167449(US9073906, 183)
Affinity DataIC50: 4.80nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167447(US9073906, 176)
Affinity DataIC50: 5nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167448(US9073906, 177)
Affinity DataIC50: 5nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384529(CHEMBL2036424 | US9073906, 2)
Affinity DataIC50: 12nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167435(US9073906, 59)
Affinity DataIC50: 14nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167446(US9073906, 175)
Affinity DataIC50: 14nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167436(US9073906, 60)
Affinity DataIC50: 17nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167439(US9073906, 89)
Affinity DataIC50: 20nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167434(US9073906, 44)
Affinity DataIC50: 79nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167442(US9073906, 124)
Affinity DataIC50: 187nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384527(CHEMBL2036422 | US9073906, 5)
Affinity DataIC50: 360nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384526(CHEMBL2036421 | US9073906, 3)
Affinity DataIC50: 363nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167432(US9073906, 14)
Affinity DataIC50: 1.66E+3nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167433(US9073906, 24)
Affinity DataIC50: 3.37E+3nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167445(US9073906, 172)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167451(US9073906, 196)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167450(US9073906, 195)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167449(US9073906, 183)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167448(US9073906, 177)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167447(US9073906, 176)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167446(US9073906, 175)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167444(US9073906, 156)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167443(US9073906, 128)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167441(US9073906, 123)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167440(US9073906, 122)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167442(US9073906, 124)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167438(US9073906, 88)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167439(US9073906, 89)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167434(US9073906, 44)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167437(US9073906, 69)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167435(US9073906, 59)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167436(US9073906, 60)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167433(US9073906, 24)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384529(CHEMBL2036424 | US9073906, 2)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM167432(US9073906, 14)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384527(CHEMBL2036422 | US9073906, 5)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

Target11-beta-hydroxysteroid dehydrogenase type 2(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandPNGBDBM50384526(CHEMBL2036421 | US9073906, 3)
Affinity DataIC50: 1.00E+4nMAssay Description:The in vitro inhibitory activities of the novel compounds to human 11β-HSD1 were evaluated in accordance with homogenous time-resolved fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent