Compile Data Set for Download or QSAR
Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 1809
LigandPNGBDBM50168297(CHEMBL3805760 | US9765060, Compound 96)
Affinity DataIC50: 0.100nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341173(US9765060, Compound 3a | (S)-2,4-diamino-6-(((5-ch...)
Affinity DataIC50: 0.300nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM50168484(CHEMBL3805137 | US9765060, Compound Y)
Affinity DataIC50: 0.400nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341228(US9765060, Compound 55 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 0.400nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341280(US9765060, Compound 107 | N-((3R,5S)-5-(5-chloro-4...)
Affinity DataIC50: 0.400nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341219(US9765060, Compound 46 | (S)-2,4-diamino-6-((1-(4-...)
Affinity DataIC50: 0.400nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341210(US9765060, Compound 37 | (S)-3-(2-(1-((2,6-diamino...)
Affinity DataIC50: 0.5nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341211(US9765060, Compound 38 | (S)-3-(2-(1-((2,6-diamino...)
Affinity DataIC50: 0.5nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341227(US9765060, Compound 54 | (S)-2,4-diamino-6-((1-(4-...)
Affinity DataIC50: 0.5nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341221(US9765060, Compound 48 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 0.5nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341270(US9765060, Compound 97 | (S)-2-(1-((2-amino-5-iodo...)
Affinity DataIC50: 0.600nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341234(US9765060, Compound 61 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 0.600nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341225(US9765060, Compound 52 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 0.700nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341239(US9765060, Compound 66 | (S)-2-amino-4-chloro-6-((...)
Affinity DataIC50: 0.700nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341226(US9765060, Compound 53 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 0.700nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341218(US9765060, Compound 45 | (S)-2,4-diamino-6-((1-(4-...)
Affinity DataIC50: 0.700nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341282(US9765060, Compound 109 | N-((3R,5S)-5-(5-chloro-3...)
Affinity DataIC50: 0.700nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341279(US9765060, Compound 106 | (S)-4-amino-6-((1-(5-chl...)
Affinity DataIC50: 0.800nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341236(US9765060, Compound 63 | (S)-4-((1-(5-(3-(2-oxa-6-...)
Affinity DataIC50: 0.800nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341235(US9765060, Compound 62 | (S)-4-((1-(5-(3-(2-oxa-6-...)
Affinity DataIC50: 0.800nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341286(US9765060, Compound 114 | N-((3R,5S)-5-(5-chloro-4...)
Affinity DataIC50: 0.900nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM50168472(CHEMBL3805348 | US9765060, Compound X)
Affinity DataIC50: 1nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341242(US9765060, Compound 69 | (S)-4-(2-(1-((2,6-diamino...)
Affinity DataIC50: 1nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM50168296(CHEMBL3805180 | US9765060, Compound 101)
Affinity DataIC50: 1nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341182(US9765060, Compound 12a | (S)-2,4-diamino-6-((cycl...)
Affinity DataIC50: 1nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341183(US9765060, Compound 13a | (S)-2,4-diamino-6-(((5-c...)
Affinity DataIC50: 1nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341248(US9765060, Compound 75 | (S)-2,4-diamino-6-(2-(3-(...)
Affinity DataIC50: 1.20nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341223(US9765060, Compound 50 | (S)-2,4-diamino-6-((1-(8-...)
Affinity DataIC50: 1.30nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341249(US9765060, Compound 76 | (S)-2,4-diamino-6-((1-(3-...)
Affinity DataIC50: 1.30nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341222(US9765060, Compound 49 | 2,4-diamino-6-(((1S)-1-(5...)
Affinity DataIC50: 1.40nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341230(US9765060, Compound 57 | (S)-2,4-diamino-6-((cyclo...)
Affinity DataIC50: 1.40nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341209(US9765060, Compound 36 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341212(US9765060, Compound 39 | (S)-3-(2-(1-((2,6-diamino...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341244(US9765060, Compound 71 | (S)-4-(2-(1-((2,6-diamino...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341180(US9765060, Compound 10a | (S)-3-(5-chloro-4-oxo-3-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341178(US9765060, Compound 8a | (S)-2-(cyclopropyl((2,6-d...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341232(US9765060, Compound 59 | (S)-2,4-diamino-6-((cyclo...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341201(US9765060, Compound 28 | (S)-2,4-diamino-6-((1-(4-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341262(US9765060, Compound 89 | (S)-2-(1-(2,6-diamino-5-c...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341267(US9765060, Compound 94 | 2,4-diamino-6-((2S,4R)-2-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341256(US9765060, Compound 83 | (S)-2,4-diamino-6-(2-(5-c...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341255(US9765060, Compound 82 | (S)-2,4-diamino-6-((1-(3-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341281(US9765060, Compound 108 | N-((3S,5S)-5-(5-chloro-4...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341278(US9765060, Compound 105 | (S)-2-amino-4-chloro-6-(...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341220(US9765060, Compound 47 | (S)-2,4-diamino-6-((1-(5-...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341245(US9765060, Compound 72 | (S)-2,4-diamino-6-(2-(3-(...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341283(US9765060, Compound 110 | N-((3R,5S)-5-(5-chloro-3...)
Affinity DataIC50: 2nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341224(US9765060, Compound 51 | (S)-2,4-diamino-6-((1-(3-...)
Affinity DataIC50: 3nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341229(US9765060, Compound 56 | (S)-2,4-diamino-6-((cyclo...)
Affinity DataIC50: 3nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

LigandPNGBDBM341243(US9765060, Compound 70 | (S)-4-(2-(1-(2,6-diamino-...)
Affinity DataIC50: 3nMAssay Description:TR-FRET monitored the formation of 3,4,5-inositol triphosphate molecule that competed with fluorescently labeled PIP3 for binding to the GRP-1 plecks...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

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