Compile Data Set for Download or QSAR
Report error Found 524 Enz. Inhib. hit(s) with all data for entry = 1840
LigandPNGBDBM343170(4-(3'-chloro-2,5'-difluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343014(4-(2,3'-dichloro-4'-fluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 7.80nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343169(4-(4'-chloro-2-fluoro-5-methoxy-3'-methyl-4-biphen...)
Affinity DataIC50: 8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342889(4-(3'-chloro-2-fluoro-5-methoxy-4-biphenylyl)-N-3-...)
Affinity DataIC50: 8.40nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343034(1-(3'-chloro-2-cyano-4'-fluoro-5-methoxy-4-bipheny...)
Affinity DataIC50: 9.20nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343040(1-(3'-chloro-2-cyano-5-methoxy-5'-methyl-4-bipheny...)
Affinity DataIC50: 11.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343041(4-(2-cyano-5-methoxy-3'-(trifluoromethyl)-4-biphen...)
Affinity DataIC50: 11.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343092(4-(3'-chloro-5-methoxy-2-methyl-4-biphenylyl)-N-3-...)
Affinity DataIC50: 12.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343046(1-(2-cyano-4'-fluoro-5-methoxy-3'-methyl-4-bipheny...)
Affinity DataIC50: 12.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343044(1-(4'-chloro-2-cyano-5-methoxy-3'-methyl-4-bipheny...)
Affinity DataIC50: 13.3nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342904(1-(2-fluoro-5-methoxy-3'-(trifluoromethyl)-4-biphe...)
Affinity DataIC50: 13.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342956(1-(3'-chloro-2-cyano-5-methoxy-5'-methyl-4-bipheny...)
Affinity DataIC50: 13.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343228(1-(2,4'-dichloro-5-methoxy-3'-methyl-4-biphenylyl)...)
Affinity DataIC50: 14nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343017(4-(2-chloro-3',5'-difluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 14.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342868(1-(3'-chloro-2-cyano-4'-fluoro-5-methoxy-4-bipheny...)
Affinity DataIC50: 14.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343068(1-(2,4'-dichloro-5-methoxy-3'-methyl-4-biphenylyl)...)
Affinity DataIC50: 15.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343168(1-(4'-chloro-2-fluoro-5-methoxy-3'-methyl-4-biphen...)
Affinity DataIC50: 16nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342905(1-(3'-chloro-2-fluoro-5-methoxy-4-biphenylyl)-N-3-...)
Affinity DataIC50: 16.3nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343110(1-(5'-chloro-2',5-dimethoxy-2-methyl-4-biphenylyl)...)
Affinity DataIC50: 16.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343022(4-(2-cyano-5-methoxy-3'-(trifluoromethyl)-4-biphen...)
Affinity DataIC50: 16.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343069(1-(2,3'-dichloro-5-methoxy-4'-methyl-4-biphenylyl)...)
Affinity DataIC50: 17.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342958(1-(4'-chloro-2-cyano-5-methoxy-3'-methyl-4-bipheny...)
Affinity DataIC50: 17.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343094(4-(5'-chloro-2',5-dimethoxy-2-methyl-4-biphenylyl)...)
Affinity DataIC50: 18.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343093(N-3-isoxazolyl-4-(5-methoxy-2-methyl-3'-(trifluoro...)
Affinity DataIC50: 18.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343038(1-(4'-chloro-2-cyano-3'-fluoro-5-methoxy-4-bipheny...)
Affinity DataIC50: 18.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343229(1-(2-chloro-3',5'-difluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 19nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342954(1-(3'-chloro-2-cyano-4'-fluoro-5-methoxy-4-bipheny...)
Affinity DataIC50: 19.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343025(4-(5-chloro-4-(5-fluoro-2-methoxy-3-pyridinyl)-2-m...)
Affinity DataIC50: 19.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343167(1-(3'-chloro-2,5'-difluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 20nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343045(1-(3'-chloro-2-cyano-5-methoxy-4'-methyl-4-bipheny...)
Affinity DataIC50: 20.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342907(1-(2-cyano-5-methoxy-3'-(trifluoromethyl)-4-biphen...)
Affinity DataIC50: 21nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343016(4-(2,4'-dichloro-5-methoxy-3'-methyl-4-biphenylyl)...)
Affinity DataIC50: 21.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343036(1-(2-cyano-3'-fluoro-5-methoxy-5'-methyl-4-bipheny...)
Affinity DataIC50: 21.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342899(1-(3'-chloro-2-cyano-5-methoxy-4-biphenylyl)-N-3-i...)
Affinity DataIC50: 21.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343132(4-(3'-chloro-2,5'-difluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 22nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343029(1-(2-cyano-5-methoxy-3'-methyl-4-biphenylyl)-N-1,3...)
Affinity DataIC50: 22.3nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343113(1-(3'-chloro-4'-fluoro-5-methoxy-2-methyl-4-biphen...)
Affinity DataIC50: 22.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342886(4-(2-fluoro-5-methoxy-3'-(trifluoromethyl)-4-biphe...)
Affinity DataIC50: 22.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343030(1-(2-cyano-3'-fluoro-5-methoxy-4'-methyl-4-bipheny...)
Affinity DataIC50: 22.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343096(4-(3'-chloro-5-methoxy-2,5'-dimethyl-4-biphenylyl)...)
Affinity DataIC50: 23.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342888(4-(4'-chloro-2-fluoro-5-methoxy-3'-methyl-4-biphen...)
Affinity DataIC50: 24nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342870(1-(3'-chloro-2-cyano-5'-fluoro-5-methoxy-4-bipheny...)
Affinity DataIC50: 24.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343097(4-(3'-chloro-4'-fluoro-5-methoxy-2-methyl-4-biphen...)
Affinity DataIC50: 25.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343031(1-(2-cyano-5-methoxy-4'-(trifluoromethyl)-4-biphen...)
Affinity DataIC50: 25.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343130(4-(3',5'-dichloro-2-fluoro-5-methoxy-4-biphenylyl)...)
Affinity DataIC50: 26nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342866(1-(4'-chloro-2-cyano-5-methoxy-3'-methyl-4-bipheny...)
Affinity DataIC50: 26.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343165(4-(2-chloro-3'-fluoro-5-methoxy-4-biphenylyl)-N-3-...)
Affinity DataIC50: 27nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM342945(US9776995, Example 299 | US9776995, Example 298 | ...)
Affinity DataIC50: 27nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343171((P)-1-(2-fluoro-5-methoxy-3''-(trifluoromethyl)-4-...)
Affinity DataIC50: 28nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

LigandPNGBDBM343208(3-amino-4-(2-chloro-3'-fluoro-5-methoxy-4-biphenyl...)
Affinity DataIC50: 28nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

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