Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 2408
LigandPNGBDBM364540(US9862711, Example 12 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 6nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364537(US9862711, Example 9 | N-(3-Hydroxy-3-methyl-butyl...)
Affinity DataIC50: 10nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364540(US9862711, Example 12 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 10nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364535(US9862711, Example 7 | Cis 3-[6-(1,3-Dimethyl-1H-p...)
Affinity DataIC50: 11nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364534(US9862711, Example 6 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 13nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364532(US9862711, Example 4 | Trans 3-[6-(1,3-Dimethyl-1H...)
Affinity DataIC50: 14nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364533(US9862711, Example 5 | Trans N-(4-Hydroxycyclohexy...)
Affinity DataIC50: 15nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364530(US9862711, Example 2 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 19nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364536(US9862711, Example 8 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 20nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364538(US9862711, Example 10 | N-(3-Hydroxy-3-methyl-buty...)
Affinity DataIC50: 20nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364529(US9862711, Example 1 | N-(3-Hydroxy-propyl)-4-meth...)
Affinity DataIC50: 22nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364538(US9862711, Example 10 | N-(3-Hydroxy-3-methyl-buty...)
Affinity DataIC50: 27nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364541(US9862711, Example 13 | Cis 3-[6-(2,5-Dimethyl-2H-...)
Affinity DataIC50: 38nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364534(US9862711, Example 6 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 40nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364541(US9862711, Example 13 | Cis 3-[6-(2,5-Dimethyl-2H-...)
Affinity DataIC50: 40nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364531(US9862711, Example 3 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 48nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364530(US9862711, Example 2 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 50nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364532(US9862711, Example 4 | Trans 3-[6-(1,3-Dimethyl-1H...)
Affinity DataIC50: 60nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364530(US9862711, Example 2 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 60nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364536(US9862711, Example 8 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 60nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364536(US9862711, Example 8 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 70nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364531(US9862711, Example 3 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 70nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364532(US9862711, Example 4 | Trans 3-[6-(1,3-Dimethyl-1H...)
Affinity DataIC50: 70nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364538(US9862711, Example 10 | N-(3-Hydroxy-3-methyl-buty...)
Affinity DataIC50: 70nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364531(US9862711, Example 3 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 80nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364539(US9862711, Example 11 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 88nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364535(US9862711, Example 7 | Cis 3-[6-(1,3-Dimethyl-1H-p...)
Affinity DataIC50: 90nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364534(US9862711, Example 6 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 90nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364533(US9862711, Example 5 | Trans N-(4-Hydroxycyclohexy...)
Affinity DataIC50: 90nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364541(US9862711, Example 13 | Cis 3-[6-(2,5-Dimethyl-2H-...)
Affinity DataIC50: 100nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364535(US9862711, Example 7 | Cis 3-[6-(1,3-Dimethyl-1H-p...)
Affinity DataIC50: 100nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364539(US9862711, Example 11 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 120nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364533(US9862711, Example 5 | Trans N-(4-Hydroxycyclohexy...)
Affinity DataIC50: 150nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364540(US9862711, Example 12 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 160nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364537(US9862711, Example 9 | N-(3-Hydroxy-3-methyl-butyl...)
Affinity DataIC50: 160nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364529(US9862711, Example 1 | N-(3-Hydroxy-propyl)-4-meth...)
Affinity DataIC50: 190nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364529(US9862711, Example 1 | N-(3-Hydroxy-propyl)-4-meth...)
Affinity DataIC50: 200nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364537(US9862711, Example 9 | N-(3-Hydroxy-3-methyl-butyl...)
Affinity DataIC50: 260nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364539(US9862711, Example 11 | Trans N-(4-Hydroxy-cyclohe...)
Affinity DataIC50: 400nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364534(US9862711, Example 6 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 450nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364535(US9862711, Example 7 | Cis 3-[6-(1,3-Dimethyl-1H-p...)
Affinity DataIC50: 630nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364532(US9862711, Example 4 | Trans 3-[6-(1,3-Dimethyl-1H...)
Affinity DataIC50: 680nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364536(US9862711, Example 8 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 680nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364530(US9862711, Example 2 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 710nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

TargetSerine/threonine-protein kinase mTOR(Human)
Novartis

US Patent
LigandPNGBDBM364534(US9862711, Example 6 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 770nMAssay Description:mTOR: Binding Assays are based on the binding and displacement of an Alexa Fluor 647-labeled, ATP-competitive kinase inhibitors to the kinase of inte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

TargetSerine/threonine-protein kinase mTOR(Human)
Novartis

US Patent
LigandPNGBDBM364532(US9862711, Example 4 | Trans 3-[6-(1,3-Dimethyl-1H...)
Affinity DataIC50: 890nMAssay Description:mTOR: Binding Assays are based on the binding and displacement of an Alexa Fluor 647-labeled, ATP-competitive kinase inhibitors to the kinase of inte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364533(US9862711, Example 5 | Trans N-(4-Hydroxycyclohexy...)
Affinity DataIC50: 1.12E+3nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

TargetSerine/threonine-protein kinase mTOR(Human)
Novartis

US Patent
LigandPNGBDBM364530(US9862711, Example 2 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 1.18E+3nMAssay Description:mTOR: Binding Assays are based on the binding and displacement of an Alexa Fluor 647-labeled, ATP-competitive kinase inhibitors to the kinase of inte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364531(US9862711, Example 3 | 3-[6-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 1.45E+3nMAssay Description:PI 3-Kinase Gamma (E), PI 3-Kinase Delta (F):The TR-FRET Adapta Universal Kinase Assay Kit was purchased from Invitrogen Corporation (Carlsbad/CA, US...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

LigandPNGBDBM364533(US9862711, Example 5 | Trans N-(4-Hydroxycyclohexy...)
Affinity DataIC50: 1.81E+3nMAssay Description:PI 3-Kinase Alpha (A), Pb 3-Kinase Beta (B), Vps34 (C), PI 4-Kinase Beta (D):The luminescence-based ATP detection reagent KinaseGlo was obtained from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2019
Entry Details
US Patent

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