Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 2632
TargetSerine/threonine-protein kinase TBK1(Human)
University of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: 440nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
University of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: 500nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
University of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: 640nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
University of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: 670nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
University of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: 770nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
University of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: 870nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
University of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: 8.76E+3nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
University of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
University of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
University of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
University of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
University of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Human)
University of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
University of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
University of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent

TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: 1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
Go to US Patent