Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 2716
TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189904(US9670201, 29 (S)-3-cyano-N-(1-methyl-3-(1-(tetrah...)
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190325(US9670201, 81 3-cyano-N-(3-((3R,4R)-1-(cyclopentan...)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189884(US9670201, 11 4-chloro-3-cyano-N-(3-(1-isobutyrylp...)
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM368656(3-cyano-N-(3-((1R,5S,8r)-3-isobutyryl-3- azabicycl...)
Affinity DataIC50: 2.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189895(US9670201, 22 (S)-3-cyano-N-(1-methyl-4-(trifluoro...)
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190346(US9670201, 95 3-cyano-N-(3-((2S,4R)-1-isobutyryl-2...)
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189905(US9670201, 30 (R)-3-cyano-4-methoxy-N-(1-methyl-4-...)
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189874(US9670201, 3 3-cyano-N-(3-(1-(cyclopentanecarbonyl...)
Affinity DataIC50: 3.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189882(US9670201, 10 3-chloro-N-(3-(1-isobutyrylpiperidin...)
Affinity DataIC50: 3.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189891(US9670201, 18 3-cyano-N-(3-(1-(2-cyclobutylacetyl)...)
Affinity DataIC50: 3.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189888(US9670201, 15 3-cyano-N-(1-methyl-3-(1-(3-methylbu...)
Affinity DataIC50: 3.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189873(US9670201, 2 3-cyano-N-(3-(1-(cyclopentanecarbonyl...)
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190324(US9670201, 80 3-cyano-N-(3-((3R,4R)-1-isobutyryl-3...)
Affinity DataIC50: 4.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189913(US9670201, 36 N-(3-(1-((1S,2R,4R)-bicyclo[2.2.1]he...)
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189918(US9670201, 41 (R)-5-chloro-N-(1,4-dimethyl-3-(1-(2...)
Affinity DataIC50: 4.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189936(US9670201, 54 (R)-3-cyano-5-hydroxy-N-(1-methyl-4-...)
Affinity DataIC50: 4.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189897(US9670201, 23 3-cyano-N-(3-(1-(cyclopentanecarbony...)
Affinity DataIC50: 4.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189879(US9670201, 7 3-cyano-N-(3-(1-isobutyrylpiperidin-4...)
Affinity DataIC50: 4.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189894(US9670201, 21 (R)-3-cyano-N-(1-methyl-4-(trifluoro...)
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189886(US9670201, 13 3-chloro-N-(3-(1-isobutyrylpiperidin...)
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190326(US9670201, 82 3-cyano-2-fluoro-N-(3-((3R,4R)-1-iso...)
Affinity DataIC50: 5.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189893(US9670201, 20 3-cyano-N-(3-(1-(2-cyclohexylacetyl)...)
Affinity DataIC50: 5.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190320(US9670201, 77 3-cyano-N-(3-((1R,5S,8r)-3-isobutyry...)
Affinity DataIC50: 5.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189890(US9670201, 17 3-cyano-N-(1-methyl-4-(trifluorometh...)
Affinity DataIC50: 5.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189881(US9670201, 9 3-cyano-4-fluoro-N-(3-(1-isobutyrylpi...)
Affinity DataIC50: 5.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189880(US9670201, 8 3-cyano-N-(3-(1-isobutyrylpiperidin-4...)
Affinity DataIC50: 5.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189906(US9670201, 31 (S)-3-cyano-4-methoxy-N-(1-methyl-4-...)
Affinity DataIC50: 5.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190312(US9670201, 70 (R)-3-cyano-N-(3-(1-isobutyryl-2,2-d...)
Affinity DataIC50: 5.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189938(US9670201, 56 (R)-3-cyano-N-(1,4-dimethyl-3-(1-(2,...)
Affinity DataIC50: 5.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189887(US9670201, 14 3-cyano-N-(3-(1-(2-cyclopentylacetyl...)
Affinity DataIC50: 5.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189910(US9670201, 34 3-cyano-N-(3-(1-(2,3-dihydro-1H-inde...)
Affinity DataIC50: 5.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190304(US9670201, 65 (R)-3-cyano-N-(3-(1-(cyclopentanecar...)
Affinity DataIC50: 5.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189878(US9670201, 6 3-cyano-N-(3-(1-isobutyrylpiperidin-4...)
Affinity DataIC50: 5.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189899(US9670201, 25 Rac-3-cyano-N-(3-(1-(2-cyclopropylpr...)
Affinity DataIC50: 5.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189898(US9670201, 24 3-cyano-N-(3-(1-(2-cyclopropylacetyl...)
Affinity DataIC50: 5.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189931(US9670201, 49 3-cyano-N-(3-(1-((1R,2S)-2-isopropyl...)
Affinity DataIC50: 6.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190317(US9670201, 74 (R)-3-cyano-N-(3-(1-(2-cyclopentylac...)
Affinity DataIC50: 6.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189902(US9670201, 27 Rac-3-cyano-N-(1-methyl-3-(1-((1R*,2...)
Affinity DataIC50: 6.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189901(US9670201, 26 Rac-3-cyano-N-(1-methyl-3-(1-((1S*,2...)
Affinity DataIC50: 6.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189933(US9670201, 51 (R)-3-cyano-N-(3-(1-(2-cyclopentylpr...)
Affinity DataIC50: 6.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189872(US9670201, 1 3-cyano-N-(3-(1-(cyclopentanecarbonyl...)
Affinity DataIC50: 7.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189903(US9670201, 28 (R)-3-cyano-N-(1-methyl-3-(1-(tetrah...)
Affinity DataIC50: 7.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189911(US9670201, 35 N-(3-(1-((1R,2S,4S)-bicyclo[2.2.1]he...)
Affinity DataIC50: 7.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190318(US9670201, 75 (R)-3-cyano-N-(3-(1-(2-cyclohexylace...)
Affinity DataIC50: 7.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190307(US9670201, 66 (R)-3-cyano-N-(3-(1-isobutyryl-2,2-d...)
Affinity DataIC50: 7.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189932(US9670201, 50 (R)-N-(3-(1-(2-(bicyclo[1.1.1]pentan...)
Affinity DataIC50: 7.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM190319(US9670201, 76 (R)-3-cyano-N-(3-(1-(2-cyclobutylace...)
Affinity DataIC50: 7.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189919(US9670201, 42 (R)-3-chloro-N-(1,4-dimethyl-3-(1-(2...)
Affinity DataIC50: 7.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189917(US9670201, 40 (R)-5-cyano-N-(1,4-dimethyl-3-(1-(2,...)
Affinity DataIC50: 7.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Pfizer

US Patent
LigandPNGBDBM189915(US9670201, 38 (R)-3-cyano-N-(1,4-dimethyl-3-(1-(2,...)
Affinity DataIC50: 7.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/4/2020
Entry Details
US Patent

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