Compile Data Set for Download or QSAR
Report error Found 129 Enz. Inhib. hit(s) with all data for entry = 2955
TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM385715(US9938222, Example 33 | Trans-2-(2-((2′-fluo...)
Affinity DataEC50:  60nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM385807(Trans-(2-((2′-fluoro-5′-isopropoxy-[1,...)
Affinity DataEC50:  60nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386968(US9938222, Example 97)
Affinity DataEC50:  70nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384313((1R,2R)-2-(((2′,3-Difluoro-5′-phenoxy-...)
Affinity DataEC50:  80nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384305((Trans)-(+/−)-2-(((2′,3-difluoro-5R...)
Affinity DataEC50:  80nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386987(US9938222, Example 116)
Affinity DataEC50:  90nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386975(US9938222, Example 104)
Affinity DataEC50:  90nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386927(US9938222, Example 58 | US9938222, Example 57 | US...)
Affinity DataEC50:  110nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386984(US9938222, Example 113)
Affinity DataEC50:  120nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386927(US9938222, Example 58 | US9938222, Example 57 | US...)
Affinity DataEC50:  120nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386971(US9938222, Example 102 | US9938222, Example 101 | ...)
Affinity DataEC50:  130nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386985(Trans-2-(((2′-fluoro-5′-((6-methylpyri...)
Affinity DataEC50:  140nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386976(US9938222, Example 105)
Affinity DataEC50:  140nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386965(US9938222, Example 94)
Affinity DataEC50:  140nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384305((Trans)-(+/−)-2-(((2′,3-difluoro-5R...)
Affinity DataEC50:  160nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386974(US9938222, Example 103)
Affinity DataEC50:  170nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386967(Trans-2-(((2′,3-difluoro-5′-(3-fluorop...)
Affinity DataEC50:  180nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386934(US9938222, Example 63)
Affinity DataEC50:  180nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386913(US9938222, Example 42)
Affinity DataEC50:  180nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386959(Trans-2-(((2′-fluoro-5′-isopropoxy-3-(...)
Affinity DataEC50:  180nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386946(US9938222, Example 75)
Affinity DataEC50:  180nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386982(Trans-2-((4-(2-chloro-5-(3-fluorophenoxy)pyridin-3...)
Affinity DataEC50:  190nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386986(US9938222, Example 115)
Affinity DataEC50:  190nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386969(US9938222, Example 98)
Affinity DataEC50:  200nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384340((1S,2R)-2-(2-(2′-Fluoro-5′-isopropoxy-...)
Affinity DataEC50:  200nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386983(US9938222, Example 112)
Affinity DataEC50:  210nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384345(Trans-2-(((2′-chloro-3-fluoro-5′-isopr...)
Affinity DataEC50:  210nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386916(US9938222, Example 45)
Affinity DataEC50:  220nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386938(US9938222, Example 67)
Affinity DataEC50:  230nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384291((METHOD A) | US9938222, Example 2)
Affinity DataEC50:  250nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386921(US9938222, Example 50)
Affinity DataEC50:  260nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386971(US9938222, Example 102 | US9938222, Example 101 | ...)
Affinity DataEC50:  260nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386978(US9938222, Example 108 | US9938222, Example 109 | ...)
Affinity DataEC50:  260nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386971(US9938222, Example 102 | US9938222, Example 101 | ...)
Affinity DataEC50:  270nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386977(US9938222, Example 106)
Affinity DataEC50:  270nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386915(US9938222, Example 44)
Affinity DataEC50:  270nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386914(US9938222, Example 43)
Affinity DataEC50:  280nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386935(US9938222, Example 64)
Affinity DataEC50:  290nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386964(Trans-2-(((5′-((R)-sec-butoxy)-2′-fluo...)
Affinity DataEC50:  300nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386963(Trans-2-(((5′-(4-Chlorophenoxy)-2′-flu...)
Affinity DataEC50:  300nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM384320(US9938222, Example 12 | US9938222, Example 14 | Tr...)
Affinity DataEC50:  310nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386917(US9938222, Example 46)
Affinity DataEC50:  310nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386933(US9938222, Example 62)
Affinity DataEC50:  310nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386962(Trans-2-(((5′-(3,4-difluorophenoxy)-2′...)
Affinity DataEC50:  310nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386978(US9938222, Example 108 | US9938222, Example 109 | ...)
Affinity DataEC50:  310nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386937(US9938222, Example 66)
Affinity DataEC50:  320nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM385620(Trans-2-(2-(2′-fluoro-5′-isopropoxy-[1...)
Affinity DataEC50:  320nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386936(US9938222, Example 65)
Affinity DataEC50:  330nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM386922(US9938222, Example 52 | US9938222, Example 53 | US...)
Affinity DataEC50:  330nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetFree fatty acid receptor 4(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM385744(Trans-(2-((2′-fluoro-5′-isopropoxy-[1,...)
Affinity DataEC50:  330nMAssay Description:For the pERK assay, 3×106 cells/mL cryopreserved human and mouse cells were thawed rapidly in a 37° C. water bath and added to a T-225 flask containi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

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