Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 10035
TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510018BDBM510018(WO2021205290, Example 27 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 0.0300nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510022BDBM510022(WO2021205290, Example 34 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 0.600nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510043BDBM510043(WO2021205290, Example 71 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 0.930nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510024BDBM510024(WO2021205290, Example 37 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 1.42nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510019BDBM510019(WO2021205290, Example 28 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 2.47nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 509969BDBM509969(WO2021205290, Example 4 | (3S)-3-({N-[(4-methoxy-1...)
Affinity DataIC50: 2.98nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510036BDBM510036(WO2021205290, Example 62 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 4.29nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510023BDBM510023(WO2021205290, Example 35 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 4.43nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510027BDBM510027(WO2021205290, Example 42 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 5.25nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510047BDBM510047(WO2021205290, Example 75 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 5.5nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510042BDBM510042(WO2021205290, Example 70 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 5.89nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510021BDBM510021(WO2021205290, Example 30 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 6.13nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510041BDBM510041(WO2021205290, Example 68 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 7.56nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510038BDBM510038(WO2021205290, Example 65 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 7.67nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510040BDBM510040(WO2021205290, Example 67 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 8.82nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510044BDBM510044(WO2021205290, Example 72 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 8.91nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510020BDBM510020(WO2021205290, Example 29 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 9.57nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510011BDBM510011(WO2021205290, Example 16 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 11nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510034BDBM510034(WO2021205290, Example 53 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 14nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510017BDBM510017(WO2021205290, Example 24 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 14nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510035BDBM510035(WO2021205290, Example 59 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 14nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510012BDBM510012(WO2021205290, Example 17 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 18nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510016BDBM510016(WO2021205290, Example 23 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 21nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 509970BDBM509970(WO2021205290, Example 9 | (3S)-3-({N-[(4-methoxy-1...)
Affinity DataIC50: 34nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510037BDBM510037(WO2021205290, Example 64 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 35nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510039BDBM510039(WO2021205290, Example 66 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 40nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510030BDBM510030(WO2021205290, Example 45 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 41nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510046BDBM510046(WO2021205290, Example 74 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 44nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510038BDBM510038(WO2021205290, Example 65 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  51nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 509971BDBM509971(WO2021205290, Example 10 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 64nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510014BDBM510014(WO2021205290, Example 19 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 65nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510013BDBM510013(WO2021205290, Example 18 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 66nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 509974BDBM509974(WO2021205290, Example 11 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 71nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510007BDBM510007(WO2021205290, Example 12 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 74nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510029BDBM510029(WO2021205290, Example 44 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 91nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510025BDBM510025(WO2021205290, Example 39 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 92nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510015BDBM510015(WO2021205290, Example 21 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 104nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510007BDBM510007(WO2021205290, Example 12 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  109nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510045BDBM510045(WO2021205290, Example 73 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 117nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510028BDBM510028(WO2021205290, Example 43 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 118nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510008BDBM510008(WO2021205290, Example 13 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 139nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510010BDBM510010(WO2021205290, Example 15 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 147nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510032BDBM510032(WO2021205290, Example 51 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 152nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510040BDBM510040(WO2021205290, Example 67 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  163nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 509971BDBM509971(WO2021205290, Example 10 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  205nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510031BDBM510031(WO2021205290, Example 48 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 255nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510026BDBM510026(WO2021205290, Example 40 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 306nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510043BDBM510043(WO2021205290, Example 71 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  315nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510009BDBM510009(WO2021205290, Example 14 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataIC50: 348nMAssay Description:Proteolytic activity of SARS-CoV-2 Coronavirus 3CL protease is measured using a continuous fluorescence resonance energy transfer assay. The SARS-CoV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

TargetReplicase polyprotein 1ab(2019-nCoV)
Pfizer

WIPO
LigandChemical structure of BindingDB Monomer ID 510009BDBM510009(WO2021205290, Example 14 | (3S)-3-({N-[(4-methoxy-...)
Affinity DataEC50:  505nMAssay Description:The ability of compounds to prevent SARS-CoV-2 coronavirus-induced cell death or cytopathic effect can be assessed via cell viability, using an assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2022
Entry Details
WIPO WO2021205290

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