Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 10360
LigandPNGBDBM530465(8-(4-Ethyl-3-(hydroxymethyl)-5-oxo-4,5-dihydro-1H-...)
Affinity DataIC50: 1.33nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530467(3-(5-Chloro-3-methyl-1H-pyrazol-4-yl)-7-fluoro-8-(...)
Affinity DataIC50: 2.10nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530464(7-Fluoro-8-(2-(2-hydroxypropan-2-yl)-1-methyl-1H-i...)
Affinity DataIC50: 2.11nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530469(7-Fluoro-8-(5-(2-hydroxypropan-2-yl)-1-methyl-1H-1...)
Affinity DataIC50: 2.51nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530466(3-(5-Chloro-3-methyl-1H-pyrazol-4-yl)-7-fluoro-8-(...)
Affinity DataIC50: 2.69nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530468(7-Fluoro-8-(2-(2-hydroxypropan-2-yl)-1-methyl-1H-i...)
Affinity DataIC50: 4.07nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530471(3-(2-Chloro-4-methylpyridin-3-yl)-7-fluoro-8-(5-(2...)
Affinity DataIC50: 13nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071

LigandPNGBDBM530470(3-(2-Chloro-4-methylpyridin-3-yl)-7-fluoro-8-(2-(2...)
Affinity DataIC50: 13nMAssay Description: To detect DHODH enzyme activities, dichloroindophenol (DCIP) is added as the final electron acceptor in the assay. DCIP can accept electrons from th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2022
Entry Details
WIPO WO2022070071