Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 10415
TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533768BDBM533768(WO2022079616, Example 1.05 | Isobutyl 5-(3-(4-carb...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533767BDBM533767(WO2022079616, Example 1.04 | 2-(Methylthio)ethyl 5...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533770BDBM533770(WO2022079616, Example 1.07 | Thiazol-5-ylmethyl 5-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533769BDBM533769(WO2022079616, Example 1.06 | 2-Methoxy-2-oxoethyl ...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533863BDBM533863(WO2022079616, Example 2.1)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533771BDBM533771(WO2022079616, Example 1.08 | 2-Morpholinoethyl 5-(...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533864BDBM533864(WO2022079616, Example 3.1 | Methyl 2-chloro-5-(N-m...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533773BDBM533773(WO2022079616, Example 1.10 | 2,2,2-Trifluoroethyl ...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533772BDBM533772(WO2022079616, Example 1.09 | Ethyl 5-(3-(4-carbamo...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533865BDBM533865(WO2022079616, Example 4.1 | Methyl 2-(3-(4-carbamo...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533775BDBM533775(WO2022079616, Example 1.12 | 2-(Dimethylamino)-2-o...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533774BDBM533774(WO2022079616, Example 1.11 | 2-Methoxyethyl 5-(3-(...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533782BDBM533782(WO2022079616, Example 1.13 | isopropyl 5-(3-(4-car...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533786BDBM533786(WO2022079616, Example 1.15 | rac-(Tetrahydrofuran-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533790BDBM533790(WO2022079616, Example 1.16 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533793BDBM533793(WO2022079616, Example 1.18 | 2-Chloro-5-(N-methyl-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533791BDBM533791(WO2022079616, Example 1.17 | t-Butyl 2-chloro-5-(N...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533812BDBM533812(WO2022079616, Example 1.19 | 2-Morpholinoethyl 2-c...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533813BDBM533813(WO2022079616, Example 1.21 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533860BDBM533860(WO2022079616, Example 1.25 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533764BDBM533764(WO2022079616, Example 1.01 | N-(4-cyanophenyl)-N-m...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533766BDBM533766(WO2022079616, Example 1.03 | 5-(3-(4-Carbamoylphen...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533861BDBM533861(WO2022079616, Example 1.26 | Methyl 5-(N-methyl-3-...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533765BDBM533765(WO2022079616, Example 1.02 | tert-Butyl 5-(3-(4-ca...)
Affinity DataIC50: 100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533862BDBM533862(WO2022079616, Example 1.27 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533793BDBM533793(WO2022079616, Example 1.18 | 2-Chloro-5-(N-methyl-...)
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533812BDBM533812(WO2022079616, Example 1.19 | 2-Morpholinoethyl 2-c...)
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533865BDBM533865(WO2022079616, Example 4.1 | Methyl 2-(3-(4-carbamo...)
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533837BDBM533837(WO2022079616, Example 1.22 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533783BDBM533783(WO2022079616, Example 1.14 | rac-1-((Ethoxycarbony...)
Affinity DataIC50: 550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533764BDBM533764(WO2022079616, Example 1.01 | N-(4-cyanophenyl)-N-m...)
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533790BDBM533790(WO2022079616, Example 1.16 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533862BDBM533862(WO2022079616, Example 1.27 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533863BDBM533863(WO2022079616, Example 2.1)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533771BDBM533771(WO2022079616, Example 1.08 | 2-Morpholinoethyl 5-(...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533864BDBM533864(WO2022079616, Example 3.1 | Methyl 2-chloro-5-(N-m...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533813BDBM533813(WO2022079616, Example 1.21 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533856BDBM533856(WO2022079616, Example 1.23 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 1.00E+3nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533837BDBM533837(WO2022079616, Example 1.22 | Methyl 2-chloro-5-(N-...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPhosphatidylinositol 4-kinase(Cryptosporidium parvum (strain Iowa II))
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533857BDBM533857(WO2022079616, Example 1.24 | Methyl 2-chloro-5-(3-...)
Affinity DataIC50: 1.00E+3nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533856BDBM533856(WO2022079616, Example 1.23 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533783BDBM533783(WO2022079616, Example 1.14 | rac-1-((Ethoxycarbony...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533857BDBM533857(WO2022079616, Example 1.24 | Methyl 2-chloro-5-(3-...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616

TargetPI3K/PI4K catalytic domain-containing protein(Cryptosporidium hominis)
Novartis

WIPO
LigandChemical structure of BindingDB Monomer ID 533860BDBM533860(WO2022079616, Example 1.25 | Methyl 5-(3-(4-carbam...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022079616