Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 11072
LigandChemical structure of BindingDB Monomer ID 582622BDBM582622(WO2023288264, Compound 14 | WO2023288264, Compound...)
Affinity DataIC50: 0.25nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582625BDBM582625(WO2023288264, Compound 17)
Affinity DataIC50: 0.300nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582633BDBM582633(WO2023288264, Compound 24)
Affinity DataIC50: 0.390nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582622BDBM582622(WO2023288264, Compound 14 | WO2023288264, Compound...)
Affinity DataIC50: 0.610nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582618BDBM582618(WO2023288264, Compound 10)
Affinity DataIC50: 1.19nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582617BDBM582617(WO2023288264, Compound 9)
Affinity DataIC50: 1.63nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582626BDBM582626(WO2023288264, Compound 18)
Affinity DataIC50: 1.65nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582630BDBM582630(WO2023288264, Compound 21)
Affinity DataIC50: 1.98nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582608BDBM582608(WO2023288264, Compound 4 | WO2023288264, Compound ...)
Affinity DataIC50: 2.34nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582623BDBM582623(WO2023288264, Compound 15)
Affinity DataIC50: 3.06nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582632BDBM582632(WO2023288264, Compound 23)
Affinity DataIC50: 3.34nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582629BDBM582629(WO2023288264, Compound 20)
Affinity DataIC50: 3.48nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582615BDBM582615(WO2023288264, Compound 8)
Affinity DataIC50: 4.73nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582621BDBM582621(WO2023288264, Compound 13)
Affinity DataIC50: 6.36nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582608BDBM582608(WO2023288264, Compound 4 | WO2023288264, Compound ...)
Affinity DataIC50: 9.23nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582628BDBM582628(WO2023288264, Compound 19)
Affinity DataIC50: 14nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582619BDBM582619(WO2023288264, Compound 11)
Affinity DataIC50: 15nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582614BDBM582614(WO2023288264, Compound 7)
Affinity DataIC50: 18nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582608BDBM582608(WO2023288264, Compound 4 | WO2023288264, Compound ...)
Affinity DataIC50: 18nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582607BDBM582607(WO2023288264, Compound 3)
Affinity DataIC50: 23nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582631BDBM582631(WO2023288264, Compound 22)
Affinity DataIC50: 24nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582634BDBM582634(WO2023288264, Compound 25)
Affinity DataIC50: 27nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582620BDBM582620(WO2023288264, Compound 12)
Affinity DataIC50: 47nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582545BDBM582545(WO2023288264, Compound 2)
Affinity DataIC50: 64nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264

LigandChemical structure of BindingDB Monomer ID 582544BDBM582544(WO2023288264, Compound 1)
Affinity DataIC50: 121nMAssay Description:Inhibitors were dissolved in 100% DMSO at a stock concentration of 10 mM. A 100X, 10-point, 4-fold serial dilution of each inhibitor was created in 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details
WIPO WO2023288264