Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 4369
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65920(2-[[1-[(5-bromo-2-fluorophenyl)methyl]-3-indolyl]s...)
Affinity DataEC50:  1.38E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65918(VU0405645-1 | cid_44475948 | 2-[4,6-difluoro-1-[[3...)
Affinity DataEC50:  1.85E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65909(cid_44216758 | N-(5-methyl-3-isoxazolyl)-2-[[1-[[3...)
Affinity DataEC50:  2.19E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65921(2-[[1-[[2-fluoro-5-(1H-pyrazol-5-yl)phenyl]methyl]...)
Affinity DataEC50:  3.07E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65915(VU0402606-1 | cid_44247544 | N-(5-methyl-1,2-oxazo...)
Affinity DataEC50:  3.21E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65914(2-[[1-[(3-bromophenyl)methyl]-3-indolyl]sulfonyl]-...)
Affinity DataEC50:  3.79E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65919(cid_44475950 | 2-[[1-[[2-fluoro-3-(1H-pyrazol-5-yl...)
Affinity DataEC50:  4.40E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65911(cid_44241485 | 2-[1-[(3-chloro-2-fluorophenyl)meth...)
Affinity DataEC50:  5.10E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65916(2-[[1-[(3-fluorophenyl)methyl]-3-indolyl]sulfonyl]...)
Affinity DataEC50:  5.22E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65917(2-[1-[(3-bromophenyl)methyl]-4,6-bis(fluoranyl)ind...)
Affinity DataEC50:  5.37E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65907(VU0366968-1 | 2-[1-[(3-chlorophenyl)methyl]indol-3...)
Affinity DataEC50:  5.82E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65908(VU0366971-1 | cid_44129593 | 2-[[1-[(3-methoxyphen...)
Affinity DataEC50:  6.54E+3nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65910(VU0404018 | 2-[[1-[(6-fluoro-3-pyridinyl)methyl]-3...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65913(2-[1-[(2-chlorophenyl)methyl]indol-3-yl]sulfonyl-N...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM65912(cid_44216757 | 2-[1-[[3-(6-chloranylpyridin-3-yl)p...)
Affinity DataEC50:  3.00E+4nMAssay Description:Assay Provider: P. Jeffery Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 Mus...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2011
Entry Details
PCBioAssay