| Assay Method Information | |
| | Scintillation Proximity Assay (SPA) |
| Description: | The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-33P]ATP. After incubation, the phosphorylated substrate was separated from nonincorporated radioactive ATP using SPA beads. Incorporated radioactivity was measured using Packard TopCount. |
| Affinity data for this assay | |
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