| Assay Method Information | |
| | Radioligand Binding Assay |
| Description: | The radioligands used were 1 nM (2R,3R,4S,5R)-2-(2-chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-3,4-diol ([3H]CCPA) for hA1, 10 nM (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-β-D-ribofuronamide) ([3H]NECA) for hA2a, and 1 nM 2-(1-hexynyl)-N6-methyladenosine [3H] ([3H]HEMADO) for hA3 receptors. |
| Affinity data for this assay | |
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