Assay Method Information

Assay Name:  ChEMBL_2202742 (CHEMBL5115450)
Description:  Inhibition of CYP2D6 in human kidney microsomes assessed as inhibition of 20-HETE formation using 3-[2-(N,N-diethyl-N-methyl-amino)ethyl]-7-methoxy-4-methyl-coumarin as substrate in presence of arachidonic acid and NADPH by fluorescence assay
Affinity data for this assay
 

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