| Assay Method Information | |
| | ChEMBL_1636028 (CHEMBL3878926) |
| Description: | Antagonist activity at human 5-HT3A expressed in HEK293 cells assessed as reduction in acetylcholine-induced activity preincubated for 30 mins followed by addition of acetylcholine measured for 2 mins by Fluo-4AM dye based FLIPR assay |
| Affinity data for this assay | |
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