Assay Method Information

Assay Name:  ChEMBL_2033572 (CHEMBL4687730)
Description:  Competitive inhibition of CYP2C9 in pooled human liver microsomes using S-warfarin as substrate preincubated for 5 mins followed by NADPH-generating system addition and measured after 20 mins by Lineweaver-Burk plot analysis
Affinity data for this assay
 

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