Assay Method Information

Assay Name:  ChEMBL_1660886 (CHEMBL4010498)
Description:  Inhibition of CYP2A6 in human liver microsomes assessed as enzyme-mediated metabolite formation using coumarin as substrate incubated for 5 mins followed by NADPH addition measured after 30 mins by LC-MS/MS analysis
Affinity data for this assay
 

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