| Assay Method Information | |
| | ChEMBL_1676974 (CHEMBL4027117) |
| Description: | Antagonist activity at rat alpha4beta2 nAChR expressed in HEK cells assessed as inhibition of epibatidine-induced membrane potential preincubated for 10 mins followed by epibatidine addition by fluorescence assay |
| Affinity data for this assay | |
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