| Assay Method Information | |
| | ChEMBL_2025080 (CHEMBL4678893) |
| Description: | Inhibition of human recombinant N-terminal GST-TEV tagged CDK12 (696 to 1082 residues)/full length human CyclinK expressed in baculovirus expression system using FITC-X-GSRTPMY-NH2 as substrate preincubated for 10 mins followed by MgCl2 addition and measured after 240 mins in presence of 5 mM ATP by mobility shift assay |
| Affinity data for this assay | |
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