Assay Method Information

Assay Name:  ChEMBL_1903851 (CHEMBL4406073)
Description:  Antagonist activity at human Gi/o-coupled D3 receptor expressed in HEK293T cells assessed as suppression of dopamine-induced inhibition of isoproterenol-stimulated cAMP accumulation preincubated for 10 mins followed by dopamine stimulation and measured after 20 mins by Glosensor-based luminescence assay
Affinity data for this assay
 

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