Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 9GTC
TargetLysosomal alpha-glucosidase(Human)
University of Toyama

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583381BDBM50583381(CHEMBL5029066 | US20230339856, Compound (IIb1))
Affinity DataKi:  19nMAssay Description:Inhibition of human GAA using 4-methylumbelliferyl-alpha-D-glucopyranoside as substrate preincubated for 45 min followed by substrate addition and me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLysosomal alpha-glucosidase(Human)
University of Toyama

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583381BDBM50583381(CHEMBL5029066 | US20230339856, Compound (IIb1))
Affinity DataKi:  6.40E+3nMAssay Description:The inhibiting activity on recombinant human acid α-glucosidase (rhGAA) of the compounds is implemented using the Fluopol-ABPP method (Fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetLysosomal alpha-glucosidase(Human)
University of Toyama

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583381BDBM50583381(CHEMBL5029066 | US20230339856, Compound (IIb1))
Affinity DataIC50: 4.91E+4nMAssay Description:The inhibiting activity on recombinant human acid α-glucosidase (rhGAA) of the compounds is implemented using the Fluopol-ABPP method (Fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
US Patent
PDB3D3D Structure (crystal)