Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 9NT7
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202222BDBM50202222(N-tert-butyl-6,7-dichloro-3-(methylsulfonyl)quinox...)
Affinity DataIC50: 32nMAssay Description:Effect on augmentation of [125]GLP1 binding to human GLP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202222BDBM50202222(N-tert-butyl-6,7-dichloro-3-(methylsulfonyl)quinox...)
Affinity DataEC50:  101nMAssay Description:Agonist activity at human GLP1 receptor expressed in BHK cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202222BDBM50202222(N-tert-butyl-6,7-dichloro-3-(methylsulfonyl)quinox...)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human GLP1 assessed as stimulation of cAMPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)