Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 9XDR
TargetKappa-type opioid receptor(Human)
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366356BDBM50366356(EMD-61753 | ASIMADOLINE HYDROCHLORIDE)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human kappa opioid receptor expressed in COS7 cells after 60 mins IP1 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366356BDBM50366356(EMD-61753 | ASIMADOLINE HYDROCHLORIDE)
Affinity DataKi:  2nMAssay Description:Affinity at K opioid receptor on membranes prepared from guinea pig cerebellum by [3H]- 69593 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article
PDB3D3D Structure (crystal)
TargetKappa-type opioid receptor(Human)
Dr. Reddy'S Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366356BDBM50366356(EMD-61753 | ASIMADOLINE HYDROCHLORIDE)
Affinity DataKi:  5.60nMAssay Description:Binding affinity to human recombinant KOR assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)