TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKd:  1.80E+3nMAssay Description:Compound was evaluated for the binding constant for association with nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataEC50:  3.20E+6nMAssay Description:In vitro ability to inhibit the binding of [125I]-alpha-bungarotoxin to nicotinic acetylcholine receptor on membranes prepared from the electric orga...More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataEC50:  200nMAssay Description:Functional potency for nAChR subtype Alpha-1-beta-1-delta gamma (torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKd:  230nMAssay Description:Compound was evaluated for the binding constant for association with nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKd:  18nMAssay Description:Compound was evaluated for the binding constant for association with nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataEC50:  6.00E+4nMAssay Description:Functional potency for nAChR subtype Alpha-1-beta-1-delta gamma(torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataEC50:  4.11E+5nMAssay Description:Functional potency for nAChR subtype Alpha1-beta1 delta gamma (torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:inhibition of (-)-[3H]nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [3H]MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of currents when compound wascoapplied with acetylcholine to recombinant Torpedo nAcChoR (from 6 oocytes)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of currents when compound wascoapplied with acetylcholine to recombinant Torpedo nAcChoR (from 6 oocytes)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  2.70nMAssay Description:Binding potency for nAChR subtype Alpha-1-beta-1-delta gamma(torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  18nMAssay Description:Binding affinity against nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  250nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Pacific electric ray)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi:  314nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  314nMAssay Description:Binding potency for nAChR subtype Alpha-1-beta-1-delta gamma(torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  331nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  370nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Pacific electric ray)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi:  384nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  550nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  690nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  3.54E+3nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  6.27E+3nMAssay Description:Inhibition of [125I]alpha-bungarotoxin binding to nicotinic acetylcholine receptor alpha1 beta gamma delta of electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding potency for nAChR subtype Alpha-1-beta-1-delta-gamma (torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Pacific electric ray)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha(Pacific electric ray)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for its ability to displace [125 I]alpha-bungarotoxin (alpha-BgT) from torpedo alpha1-beta1-gamma1 electroplaxMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding potency for nAChR subtype Alpha-1-beta-1-delta gamma(torpedo)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  2.80E+4nMAssay Description:Binding affinity against nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  5.00E+4nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: <1.00E+5nMAssay Description:Displacement of (+/-)-[3H]epibatidine from muscle type nAChR of Torpedo californica in hepes bufferMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  3.70E+5nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  4.20E+5nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  8.30E+5nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  8.30E+6nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  3.10E+6nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  3.30E+6nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Pacific electric ray)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi:  3.10E+6nMAssay Description:Compound was evaluated for inhibition of [3H]TCP binding to Nicotinic acetylcholine receptor of Torpedo californicaMore data for this Ligand-Target Pair
 
 	

 3D Structure (crystal)
3D Structure (crystal)

































