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Report error Found 858 for UniProtKB: P30560
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKd:  0.0400nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKd:  0.0540nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350866(CHEMBL1819441)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50108501(2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimet...)
Affinity DataKi:  0.102nMAssay Description:Evaluated for the binding affinity towards Vasopressin V1a receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350852(CHEMBL1817706)
Affinity DataEC50:  0.105nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.110nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.120nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350876(CHEMBL1819542)
Affinity DataEC50:  0.123nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350869(CHEMBL1817704)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.130nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKd:  0.150nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]AVP on rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.160nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350853(CHEMBL1817707)
Affinity DataEC50:  0.162nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.180nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.180nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50166224(Vasopressin Analogue | CHEMBL410567)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against rat vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.182nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKd:  0.182nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKd:  0.190nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.200nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.240nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350851(CHEMBL1817705)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038604(3-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)
Affinity DataKi:  0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350872(CHEMBL1817761)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50008097([2-({1-[19-Amino-13-(4-azido-benzyl)-10-(2-carbamo...)
Affinity DataKd:  0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50008097([2-({1-[19-Amino-13-(4-azido-benzyl)-10-(2-carbamo...)
Affinity DataKd:  0.330nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM85096(NSC_105077 | CAS_105077 | d(CH2)5Tyr(Me)AVP)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50008097([2-({1-[19-Amino-13-(4-azido-benzyl)-10-(2-carbamo...)
Affinity DataKd:  0.331nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50008097([2-({1-[19-Amino-13-(4-azido-benzyl)-10-(2-carbamo...)
Affinity DataKd:  0.331nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350849(CHEMBL1817702)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350865(CHEMBL1819440)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  0.460nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  0.470nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.479nMAssay Description:Negative log of Kd.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.480nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  0.480nMAssay Description:Displacement of [3H]AVP from V1A receptor in Wistar rat liver membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350864(CHEMBL1819439)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350870(CHEMBL1817709)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.600nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKd:  0.603nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50350871(CHEMBL1817756)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.620nMAssay Description:Evaluated for the binding affinity towards Vasopressin V1a receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKd:  0.640nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
Upr 9023 Cnrs

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKd:  0.646nMAssay Description:Negative log of Kd.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
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