Compile Data Set for Download or QSAR
Report error Found 9 of affinity data for UniProtKB/TrEMBL: P89582
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50062551(Dolutegravir | GSK1349572 | CHEBI:76010 | S-349572)
Affinity DataEC50:  2.30nMAssay Description:Inhibition of wild type HIV-2 ROD9 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056908(3,4-di-O-caffeoylquinicacid | (1R,3R,4S,5R)-3,4-bi...)
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration of compound against strand transfer of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056908(3,4-di-O-caffeoylquinicacid | (1R,3R,4S,5R)-3,4-bi...)
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration of compound against 3'-processing of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM506(3-({4-[bis(4-hydroxy-2-oxo-2H-chromen-3-yl)methyl]...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against HIV-2 Integrase was measured using 3'-processing (3'-proc) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056938(NSC-66209 | cid_72721 | CHEMBL175266 | 2,6,7-Trihy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration of compound against strand transfer of of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056924(NSC-324362 | 3,4,5,N-Tetrahydroxy-benzamide | CHEM...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory concentration of compound against 3' processing of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056924(NSC-324362 | 3,4,5,N-Tetrahydroxy-benzamide | CHEM...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory concentration of compound against strand transfer of HIV- integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056938(NSC-66209 | cid_72721 | CHEMBL175266 | 2,6,7-Trihy...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration of compound against 3'-processing of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus 2)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50056937(3,4-dihydroxy-5-(3,4,5-trihydroxybenzoyloxy)benzoi...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration of compound against 3'-processing of HIV-2 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed