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TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM301689(US10131692, Compound 21)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205305(d[Arg4]AVP | CHEMBL375324)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205304(dVDAVP | CHEMBL435323)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205300(d[Val4]AVP | CHEMBL221436)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35709(YM-35278)
Affinity DataKi:  0.400nM ΔG°:  -53.3kJ/molepH: 7.4 T: 2°CAssay Description:The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.770nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]AVP on rat kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50078656(N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against arginine vasopressin V2 receptor using [3H]AVP as radioligand in rat adrenal medullaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50125101(Biphenyl-2-carboxylic acid [4-(1,3,4,5-tetrahydro-...)
Affinity DataIC50: 1nMAssay Description:Binding affinity towards V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against arginine vasopressin V2 receptor using [3H]AVP as radioligand in rat adrenal medullaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50078652(N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  1.20nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50087550(Biphenyl-2-carboxylic acid [3-chloro-4-(5,6,7,8-te...)
Affinity DataIC50: 1.20nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35723(N-[4-(7-Chloro-5-hydroxy-2,3,4,5-tetrahydro-benzo[...)
Affinity DataKi:  1.33nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKd:  1.5nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065124(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [3H]AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50087541(Biphenyl-2-carboxylic acid [4-(5H,11H-benzo[e]pyrr...)
Affinity DataIC50: 1.5nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50078660(N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50038601(4-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50078651(N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.80nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205296(d[Arg4,Dab8]VP | CHEMBL385739)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM85094(NSC_64759 | CAS_62357-86-2 | dDAVP)
Affinity DataKi:  1.93nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [3H]AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor of rat kidney medulla.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 2.30nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50087552(Biphenyl-2-carboxylic acid [4-(5H,11H-benzo[e]pyrr...)
Affinity DataIC50: 2.60nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)
Affinity DataKi:  3nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50075816(Mca1,D-Trp2,Sar7AVT | CHEMBL264208)
Affinity DataKd:  3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50078654(N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of (P[3H]-AVP binding towards isolated rat kidney medullary Vasopre ssin V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065110(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V2 receptor using [3H]AVP as radioligand in rat adrenal medullaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V2 receptor using [3H]AVP as radioligand in rat adrenal medullaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AVP from V2 receptor in Wistar rat kidney membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM85095(CONIVAPTAN | NSC_151171 | CAS_151171 | YM087)
Affinity DataKi:  3.04nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205292(d[Arg4,Orn8]VP | CHEMBL385068)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065110(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 3.10nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205313(d[Leu4]AVP | CHEMBL265859)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50065110(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor of rat kidney medulla.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50087543(Biphenyl-2-carboxylic acid [4-(2-chloro-5,6,7,8-te...)
Affinity DataIC50: 3.20nMAssay Description:In vitro for its binding affinity to rat V2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  3.23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205311(d[Orn4]AVP | CHEMBL375096)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205298(d[Arg4,Lys8]VP | CHEMBL375325)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
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