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TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295699(2-(3-Guanidino-propoxy)-N-(6-phenoxy-benzothiazol-...)
Affinity DataEC50:  3.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304185(2-(5-Guanidino-octanamido)-5-(3-guanidinopropoxy)-...)
Affinity DataEC50:  1.30E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304184(2-(5-Guanidinohexanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304183(2-(5-Guanidinopentanamido)-5-(3-guanidinopropoxy)-...)
Affinity DataEC50:  1.16E+5nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304182(5-(4-Aminobutoxy)-2-(8-aminooctanamido)-N-(4-pheno...)
Affinity DataEC50:  9.00E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304181(5-(4-Aminobutoxy)-2-(6-aminohexanamido)-N-(4-pheno...)
Affinity DataEC50:  9.90E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304180(2-(8-Aminooctanamido)-5-(3-aminopropoxy)-N-(4-phen...)
Affinity DataEC50:  7.20E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295707(2-(3-(4-((2,2-diphenylethylamino)methyl)phenoxy)pr...)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295706(3-{4-[(2,2-Diphenyl-ethylamino)-methyl]-phenoxy}-p...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295705(2-(3-(4-((benzhydrylamino)methyl)phenoxy)propyl)gu...)
Affinity DataEC50:  2.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295704(3-{4-[(Benzhydryl-amino)-methyl]-phenoxy}-propylam...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295703(2-(3-(4-((4-phenoxyphenylamino)methyl)phenoxy)prop...)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295702([4-(3-Amino-propoxy)-benzyl]-(4-phenoxy-phenyl)-am...)
Affinity DataEC50:  3.40E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295701(N-(3-{4-[(6-Phenoxy-benzothiazol-2-ylamino)-methyl...)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295700([4-(3-Amino-propoxy)-benzyl]-(6-phenoxy-benzothiaz...)
Affinity DataEC50:  7.60E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295698(2-(3-Amino-propoxy)-N-(6-phenoxy-benzothiazol-2-yl...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295697(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  1.78E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295696(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  3.08E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295695(2-(3-aminopropoxy)-N-(4-(3-aminopropoxy)benzyl)-N-...)
Affinity DataEC50:  3.18E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304186(2-(5-Guanidinohexanamido)-5-(3-guanidinobutoxy)-N-...)
Affinity DataEC50:  1.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304187(2-(5-Guanidino-octanamido)-5-(3-guanidinobutoxy)-N...)
Affinity DataEC50:  1.50E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304188(2-(8-Guanidinooctanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304189(N-(4-(4-Fluorophenoxy)phenyl)-2-(8-guanidinooctana...)
Affinity DataEC50:  6.00E+3nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304190(2-(5-Aminopentanamido)-5-(3-aminopropoxy)-N-(4-phe...)
Affinity DataEC50:  7.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304191(2-(6-Aminohexanamido)-5-(3-aminopropoxy)-N-(4-phen...)
Affinity DataEC50:  1.07E+5nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295697(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  5.70E+3nMAssay Description:Displacement of [125I]GVIA from rat brain membrane Cav2.2 after 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295695(2-(3-aminopropoxy)-N-(4-(3-aminopropoxy)benzyl)-N-...)
Affinity DataEC50:  5.40E+3nMAssay Description:Displacement of [125I]GVIA from rat brain membrane Cav2.2 after 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50386813(CHEMBL2047726)
Affinity DataIC50: 40.7nMAssay Description:Inhibition of rat Cav2.2 expressed in HEK293 cells under inactivating depolarizing conditions at holding potential of -115mV and stepped to 0 mV once...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50386813(CHEMBL2047726)
Affinity DataIC50: 41nMAssay Description:Inhibition of rat Cav2.2 expressed in HEK293 cells under inactivating depolarizing conditions at holding potential of -115mV and stepped to 0 mV once...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50481859(CHEMBL1088309)
Affinity DataIC50: 50nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481859(CHEMBL1088309)
Affinity DataIC50: 50nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50017702(cid_6365505 | 1-(bis(4-fluorophenyl)methyl)-4-cinn...)
Affinity DataIC50: 80nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481862(CHEMBL1087275)
Affinity DataIC50: 90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50095765(1-[Bis-(4-fluoro-phenyl)-methyl]-4-(2,3,4-trimetho...)
Affinity DataIC50: 90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481860(CHEMBL1087660)
Affinity DataIC50: 90nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50461289(Z160 | MK-6721 | NMED-160 | NP-118809 | Z-160)
Affinity DataIC50: 110nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481858(CHEMBL1086621)
Affinity DataIC50: 110nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481868(CHEMBL1088610)
Affinity DataIC50: 130nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481864(CHEMBL1087237)
Affinity DataIC50: 150nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481466(CHEMBL599217)
Affinity DataIC50: 150nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481863(CHEMBL1088464)
Affinity DataIC50: 190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481861(CHEMBL1087779)
Affinity DataIC50: 190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481869(CHEMBL1088308)
Affinity DataIC50: 190nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
LigandPNGBDBM50481449(CHEMBL599408)
Affinity DataIC50: 260nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50438747(CHEMBL2414787)
Affinity DataIC50: 340nMAssay Description:Inhibition of rat N-type Cav2.2 channel expressed in HEK293 cells under hyperpolarized condition by whole cell patch-clamp manual electrophysiology a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50481867(CHEMBL1088174)
Affinity DataIC50: 540nMAssay Description:Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50434732(CHEMBL2385364)
Affinity DataIC50: 850nMAssay Description:Inhibition of rat brain Cav2.2 N-type channel expressed in HEK cells after 20 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50438746(CHEMBL2414771)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat N-type Cav2.2 channel expressed in HEK293 cells under depolarized condition by whole cell patch-clamp manual electrophysiology assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50117922(CHEMBL45816 | Methoxy-acetic acid 2-(2-{[3-(1H-ben...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat Cav2.2-alpha1beta/beta3 expressed in HEK293 cells assessed as decrease in calcium mobilization response to KCl after 1 hr by Fluo-4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rat)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50434737(CHEMBL2385359)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of rat brain Cav2.2 N-type channel expressed in HEK cells after 20 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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