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Report error Found 22 of affinity data for UniProtKB/TrEMBL: W8NX99
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192658(N’-(2-nitrophenylmethylene)benzohydrazide (1i...)
Affinity DataKi:  4.20nM ΔG°:  -49.7kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
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Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192660(N’-(4-nitrophenylmethylene)benzohydrazide (1k...)
Affinity DataKi:  5.53nM ΔG°:  -49.0kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192659(N’-(3-nitrophenylmethylene)benzohydrazide (1j...)
Affinity DataKi:  5.86nM ΔG°:  -48.9kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192654(N’-(4-chlorophenylmethylene)benzohydrazide (1...)
Affinity DataKi:  6.34nM ΔG°:  -48.7kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192652(N’-(2-chlorophenylmethylene)benzohydrazide (1...)
Affinity DataKi:  7.30nM ΔG°:  -48.3kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192655(N’-(2-methoxyphenylmethylene)benzohydrazide (...)
Affinity DataKi:  8.14nM ΔG°:  -48.0kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192653(N’-(3-chlorophenylmethylene)benzohydrazide (1...)
Affinity DataKi:  8.63nM ΔG°:  -47.9kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192650(N’-(phenylmethylene)benzohydrazide (1a))
Affinity DataKi:  13nM ΔG°:  -46.8kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192657(N’-(4-methoxyphenylmethylene)benzohydrazide (...)
Affinity DataKi:  19.8nM ΔG°:  -45.7kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192656(N’-(3-methoxyphenylmethylene)benzohydrazide (...)
Affinity DataKi:  28.6nM ΔG°:  -44.8kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192668(2-phenyl-5-(4-nitrophenyl)-1,3,4-oxadiazole (2k))
Affinity DataKi:  47.3nM ΔG°:  -43.5kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192667(2-phenyl-5-(2-nitrophenyl)-1,3,4-oxadiazole (2i))
Affinity DataKi:  57nM ΔG°:  -43.0kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM63525(MLS000709882 | SMR000287045 | cid_577329 | 2-(3-ni...)
Affinity DataKi:  63.4nM ΔG°:  -42.7kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM48184(cid_259755 | MLS000108072 | SMR000104035 | 2-(3-ch...)
Affinity DataKi:  70.2nM ΔG°:  -42.5kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192662(2-phenyl-5-(2-chlorophenyl)-1,3,4-oxadiazole (2c))
Affinity DataKi:  92.1nM ΔG°:  -41.8kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192651(N’-(4-methylphenylmethylene)benzohydrazide (1...)
Affinity DataKi:  95.9nM ΔG°:  -41.7kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192663(2-phenyl-5-(4-chlorophenyl)-1,3,4-oxadiazole (2e))
Affinity DataKi:  99.3nM ΔG°:  -41.6kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192661(2,5-diphenyl-1,3,4-oxadiazole (2a))
Affinity DataKi:  124nM ΔG°:  -41.0kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192665(2-phenyl-5-(3-methoxyphenyl)-1,3,4-oxadiazole (2g))
Affinity DataKi:  144nM ΔG°:  -40.6kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192664(2-phenyl-5-(2-methoxyphenyl)-1,3,4-oxadiazole (2f))
Affinity DataKi:  216nM ΔG°:  -39.6kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM192666(2-phenyl-5-(4-methoxyphenyl)-1,3,4-oxadiazole (2h))
Affinity DataKi:  337nM ΔG°:  -38.4kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed
TargetCathepsin L(Goat)
Kurukshetra University

LigandPNGBDBM49356(cid_259997 | SMR000118227 | MLS000120832 | 2-(4-me...)
Affinity DataKi:  1.36E+3nM ΔG°:  -34.8kJ/molepH: 5.0 T: 2°CAssay Description:The proteolytic activity was estimated at pH 5.0, 37 °C using 0.1 M acetate buffer as the incubation medium. The homogenate prepared above was incuba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2016
Entry Details Article
PubMed