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6 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Tryptophan-containing dipeptide derivatives as potent PPARgamma antagonists: design, synthesis, biological evaluation, and molecular modeling.EBI
Graduate School of The Chinese Academy of Sciences
Pyrazolidine-3,5-dione derivatives as potent non-steroidal agonists of farnesoid X receptor: virtual screening, synthesis, and biological evaluation.EBI
Graduate School of The Chinese Academy of Sciences
Synthesis and evaluation of a series of benzopyran derivatives as PPAR alpha/gamma agonists.EBI
Graduate School of The Chinese Academy of Sciences
Sequence-based design and discovery of peptide inhibitors of HIV-1 integrase: insight into the binding mode of the enzyme.EBI
Graduate School of The Chinese Academy of Sciences
Discovery of a novel nonphosphorylated pentapeptide motif displaying high affinity for Grb2-SH2 domain by the utilization of 3'-substituted tyrosine derivatives.EBI
Graduate School of The Chinese Academy of Sciences
Identification of potent type I MetAP inhibitors by simple bioisosteric replacement. Part 1: Synthesis and preliminary SAR studies of thiazole-4-carboxylic acid thiazol-2-ylamide derivatives.EBI
Graduate School of The Chinese Academy of Sciences