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21 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of SMP-304, a novel benzylpiperidine derivative with serotonin transporter inhibitory activity and 5-HTEBI
Sumitomo Dainippon Pharma
Discovery of dihydroquinazolinone derivatives as potent, selective, and CNS-penetrant M(1) and M(4) muscarinic acetylcholine receptors agonists.EBI
Sumitomo Dainippon Pharma
Three-dimensional rational approach to the discovery of potent substituted cyclopropyl urea soluble epoxide hydrolase inhibitors.EBI
Sumitomo Dainippon Pharma
Discovery of 3H-imidazo[4,5-c]quinolin-4(5H)-ones as potent and selective dipeptidyl peptidase IV (DPP-4) inhibitors: use of a carboxylate prodrug to improve bioavailability.EBI
Sumitomo Dainippon Pharma
Dihydropyrrolo[2,3-d]pyrimidines: Selective Toll-Like Receptor 9 Antagonists from Scaffold Morphing Efforts.EBI
Sumitomo Dainippon Pharma
Synthesis, structure-activity relationships and biological evaluation of 4,5,6,7-tetrahydropyrazolopyrazines as metabotropic glutamate receptor 5 negative allosteric modulators.EBI
Sumitomo Dainippon Pharma
Discovery of DSP-1053, a novel benzylpiperidine derivative with potent serotonin transporter inhibitory activity and partial 5-HTEBI
Sumitomo Dainippon Pharma
Synthesis and optimization of 4,5,6,7-tetrahydrooxazolo[4,5-c]pyridines as potent and orally-active metabotropic glutamate receptor 5 negative allosteric modulators.EBI
Sumitomo Dainippon Pharma
Compounds and methods for inhibiting CYP26 enzymesBDB
Queens University At Kingston
Chemical compoundsBDB
Astrazeneca
JAK kinase inhibitor compounds for treatment of respiratory diseaseBDB
Theravance Biopharma R&D Ip
Benzolactam compounds as protein kinase inhibitorsBDB
Otsuka Pharmaceutical
1H-pyrazolo[4,3-b]pyridines as PDE1 inhibitorsBDB
H. Lundbeck
Bruton's tyrosine kinase inhibitorsBDB
Zibo Biopolar Changsheng Pharmaceutical
Aryldiazepine derivatives as RSV inhibitorsBDB
Enanta Pharmaceuticals
Piperidin-4-yl azetidine derivatives as JAK1 inhibitorsBDB
Incyte Holdings
Fused tricyclic compounds as Raf kinase inhibitorsBDB
Beigene
Effects of isoform-selective phosphatidylinositol 3-kinase inhibitors on osteoclasts: actions on cytoskeletal organization, survival, and resorption.BDB
Western University
Substituted phenyl hexahydropyrano[3,4-d][1,3]thiazin-2-amine compoundsBDB
Pfizer
S1P receptors modulatorsBDB
Akaal Pharma