21 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Discovery of SMP-304, a novel benzylpiperidine derivative with serotonin transporter inhibitory activity and 5-HT

Sumitomo Dainippon Pharma
Discovery of dihydroquinazolinone derivatives as potent, selective, and CNS-penetrant M(1) and M(4) muscarinic acetylcholine receptors agonists.

Sumitomo Dainippon Pharma
Three-dimensional rational approach to the discovery of potent substituted cyclopropyl urea soluble epoxide hydrolase inhibitors.

Sumitomo Dainippon Pharma
Discovery of 3H-imidazo[4,5-c]quinolin-4(5H)-ones as potent and selective dipeptidyl peptidase IV (DPP-4) inhibitors: use of a carboxylate prodrug to improve bioavailability.

Sumitomo Dainippon Pharma
Dihydropyrrolo[2,3-d]pyrimidines: Selective Toll-Like Receptor 9 Antagonists from Scaffold Morphing Efforts.

Sumitomo Dainippon Pharma
Synthesis, structure-activity relationships and biological evaluation of 4,5,6,7-tetrahydropyrazolopyrazines as metabotropic glutamate receptor 5 negative allosteric modulators.

Sumitomo Dainippon Pharma
Discovery of DSP-1053, a novel benzylpiperidine derivative with potent serotonin transporter inhibitory activity and partial 5-HT

Sumitomo Dainippon Pharma
Synthesis and optimization of 4,5,6,7-tetrahydrooxazolo[4,5-c]pyridines as potent and orally-active metabotropic glutamate receptor 5 negative allosteric modulators.

Sumitomo Dainippon Pharma
Compounds and methods for inhibiting CYP26 enzymes

Queens University At Kingston
Chemical compounds

Astrazeneca
JAK kinase inhibitor compounds for treatment of respiratory disease

Theravance Biopharma R&D Ip
Benzolactam compounds as protein kinase inhibitors

Otsuka Pharmaceutical
1H-pyrazolo[4,3-b]pyridines as PDE1 inhibitors

H. Lundbeck
Bruton's tyrosine kinase inhibitors

Zibo Biopolar Changsheng Pharmaceutical
Aryldiazepine derivatives as RSV inhibitors

Enanta Pharmaceuticals
Piperidin-4-yl azetidine derivatives as JAK1 inhibitors

Incyte Holdings
Fused tricyclic compounds as Raf kinase inhibitors

Beigene
Effects of isoform-selective phosphatidylinositol 3-kinase inhibitors on osteoclasts: actions on cytoskeletal organization, survival, and resorption.

Western University
Substituted phenyl hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds

Pfizer
S1P receptors modulators

Akaal Pharma