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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 728K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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10 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of resveratrol derivatives as novel LSD1 inhibitors: Design, synthesis and their biological evaluation.EBI
Xinxiang Medical University
Discovery of potent and novel dual NAMPT/BRD4 inhibitors for efficient treatment of hepatocellular carcinoma.EBI
Xinxiang Medical University
Discovery of novel, potent, and orally bioavailable HDACs inhibitors with LSD1 inhibitory activity for the treatment of solid tumors.EBI
Xinxiang Medical University
A comprehensive review of BET-targeting PROTACs for cancer therapy.EBI
Xinxiang Medical University
Research progress of dual inhibitors targeting crosstalk between histone epigenetic modulators for cancer therapy.EBI
Xinxiang Medical University
Recent advances in combretastatin A-4 codrugs for cancer therapy.EBI
Xinxiang Medical University
Design, synthesis, and biological evaluation of novel dual inhibitors targeting lysine specific demethylase 1 (LSD1) and histone deacetylases (HDAC) for treatment of gastric cancer.EBI
Xinxiang Medical University
Design, synthesis and in vitro evaluation of stilbene derivatives as novel LSD1 inhibitors for AML therapy.EBI
Xinxiang Medical University
Design and synthesis of tranylcypromine derivatives as novel LSD1/HDACs dual inhibitors for cancer treatment.EBI
Xinxiang Medical University
Discovery of a low-systemic-exposure DGAT-1 inhibitor with a picolinoylpyrrolidine-2-carboxylic acid moiety.EBI
Xinxiang Medical University