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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
MLN8054 and Alisertib (MLN8237): Discovery of Selective Oral Aurora A Inhibitors.EBI
Takeda Pharmaceutical
Design, synthesis and bioevaluation of N-trisubstituted pyrimidine derivatives as potent aurora A kinase inhibitors.EBI
Sun Yat-Sen University
Antitumor activity of MLN8054, an orally active small-molecule inhibitor of Aurora A kinase.EBI
Millennium Pharmaceuticals
Discovery of 2-(Anilino)pyrimidine-4-carboxamides as Highly Potent, Selective, and Orally Active Glycogen Synthase Kinase-3 (GSK-3) Inhibitors.EBI
Biocon-Bristol Myers Squibb Research and Development Center
Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 Inhibitors.EBI
Bristol-Myers Squibb Research & Development
Design, Structure-Activity Relationships, and In Vivo Evaluation of Potent and Brain-Penetrant Imidazo[1,2-EBI
Biocon-Bristol Myers Squibb Research and Development Center
Design, synthesis, biological evaluation of 6-(2-amino-1H-benzo[d]imidazole-6-yl)quinazolin-4(3H)-one derivatives as novel anticancer agents with Aurora kinase inhibition.EBI
The Key Laboratory of Chemistry For Natural Products of Guizhou Province and Chinese Academy of Sciences
Synthesis and identification of 2,4-bisanilinopyrimidines bearing 2,2,6,6-tetramethylpiperidine-N-oxyl as potential Aurora A inhibitors.EBI
Lanzhou University
MU opioid receptor modulatorsBDB
University of California
Insulin sensitisers and methods of treatmentBDB
Naia Metabolic
Imidazothiadiazole and imidazopyridazine derivatives as protease activated receptor 4 (PAR4) inhibitors for treating platelet aggregationBDB
Bristol-Myers Squibb
Structure-guided development of specific pyruvate dehydrogenase kinase inhibitors targeting the ATP-binding pocket.BDB
University of Texas Southwestern Medical Center