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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 708K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Carboxylate bioisosteres of gabapentin.EBI
Pfizer
Identification and synthesis of [1,2,4]triazolo[3,4-a]phthalazine derivatives as high-affinity ligands to the alpha 2 delta-1 subunit of voltage gated calcium channel.EBI
Merck Research Laboratories
Pyrazolopyridazine alpha-2-delta-1 ligands for the treatment of neuropathic pain.EBI
Glaxosmithkline
Rational Multitargeted Drug Design Strategy from the Perspective of a Medicinal Chemist.EBI
Shandong University
Structure-activity relationships of alpha-amino acid ligands for the alpha2delta subunit of voltage-gated calcium channels.EBI
Abbott Laboratories
Expedited SAR study of high-affinity ligands to the alpha(2)delta subunit of voltage-gated calcium channels: Generation of a focused library using a solution-phase Sn2Ar coupling methodology.EBI
Merck Research Laboratories
N-Acridin-9-yl-butane-1,4-diamine derivatives: high-affinity ligands of the alpha2delta subunit of voltage gated calcium channels.EBI
Merck Research Laboratories
Synthesis and biological evaluation of 6-aryl-6H-pyrrolo[3,4-d]pyridazine derivatives: high-affinity ligands to the alpha 2 delta subunit of voltage gated calcium channels.EBI
Merck Research Laboratories
Piperazinyl Bicyclic Derivatives as Selective Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels.EBI
Welab Barcelona
Bicyclic Diazepinones as Dual Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels and the Norepinephrine Transporter.EBI
Esteve Pharmaceuticals
SPIROCYCLIC MODULATORS OF CHOLESTEROL BIOSYNTHESIS AND THEIR USE FOR PROMOTING REMYELINATIONBDB
Genentech
1-cyano-pyrrolidine compounds as USP30 inhibitorsBDB
Mission Therapeutics
Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of disorders related theretoBDB
Arena Pharmaceuticals
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.BDB
Institut Pasteur Korea