16 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
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Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH
Takeda Pharmaceutical
Rational design of triazololipopeptides analogs of kisspeptin inducing a long-lasting increase of gonadotropins.
Umr7247
Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.
Takeda Pharmaceutical
Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.
Takeda Pharmaceutical
Trypsin resistance of a decapeptide KISS1R agonist containing an N¿-methylarginine substitution.
Takeda Pharmaceutical
Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.
Takeda Pharmaceutical
2-acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats.
Takeda Pharmaceutical
Synthesis and structure-activity relationships of 2-acylamino-4,6-diphenylpyridine derivatives as novel antagonists of GPR54.
Takeda Pharmaceutical
SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54.
Kyoto University
Metastin (KiSS-1) mimetics identified from peptide structure-activity relationship-derived pharmacophores and directed small molecule database screening.
University of Minnesota Health Science Center
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Research Triangle Institute
A new class of pentapeptide KISS1 receptor agonists with hypothalamic-pituitary-gonadal axis activation.
Takeda Pharmaceutical
Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
Array Biopharma